| Cat.No. | Name | Information |
|---|---|---|
| M2030 | Apremilast | Apremilast is a novel, orally available small molecule inhibitor of PDE4 with IC50 of 74 nM. Apremilast inhibits TNF-α release by lipopolysaccharide (LPS) with an IC50 of 104 nM. |
| M6804 | IBMX | IBMX is a pDE inhibitor (non-selective) with IC50 values of 6.5±1.2, 26.3±3.9 and 31.7±5.3 μM for PDE3, 4 and 5 respectively. |
| M56754 | Thioquinapiperifil | Thioquinapiperifil (KF31327 free base), a potent, selective and non-competitive phosphodiesterase-5 (PDE-5, IC50 of 0.074 nM) inhibitor, is used for sexual enhancement study. |
| M56753 | Lodenafil carbonate | Lodenafil carbonate, a dimer that acts as a proagent delivering Lodenafil in vivo, is an orally active phosphodiesterase type 5 (PDE5) inhibitor for the treatment of erectile dysfunction (ED). |
| M56752 | Etazolate hydrochloride | Etazolate hydrochloride (SQ 20009) is an orally active, selective inhibitor of type 4 phosphodiesterase (PDE4) with an IC50 of 2 μM. |
| M56751 | Thioquinapiperifil dihydrochloride | Thioquinapiperifil dihydrochloride (KF31327), a potent, selective and non-competitive phosphodiesterase-5 (PDE-5, IC50 of 0.074 nM) inhibitor, is used for sexual enhancement study. |
| M55688 | PF-04671536 | PF-04671536 is a highly potent and selective inhibitor of phosphodiesterase 8B (PDE8B) phosphodiesterase 8A (PDE8A). In primary human pancreatic islets, PF-04671536 increases insulin secretion in a glucose-dependent manner. |
| M49421 | ME-3183 | ME-3183 is an oral selective PDE4 inhibitor with anti-inflammatory activity for studies related to plaque psoriasis. |
| M49420 | ART-648 | ART-648 is a PDE4 inhibitor that may be used in studies related to non-alcoholic steatohepatitis. |
| M49402 | (E/Z)-HA155 | (E/Z)-HA155 is a potent Autotaxin (ATX) type I inhibitor for studies related to cancer, fibrous disorders, inflammation, pain and angiogenesis. |
| M49401 | Autotaxin-IN-3 | Autotaxin-IN-3 is an Autotaxin(ATX) inhibitor with an IC50 value of 2.4 nM. |
| M49400 | HA155 | HA155 is a potent and selective ATX inhibitor with an IC50 value of 5.7 nM. |
| M49398 | ATX inhibitor 5 | ATX inhibitor 5 is a potent, orally active inhibitor of Autotaxin (ATX) with an IC50 of 15.3 nM.Additionally, AATX inhibitor 5 exhibits anti-hepatic fibrosis activity and significantly reduces CCl4-induced hepatic fibrosis. |
| M49394 | BBT-877 | BBT-877 is an oral small molecule autotaxin (ATX) inhibitor for use in studies related to non-alcoholic steatohepatitis (NASH) and idiopathic pulmonary fibrosis (IPF). |
| M44885 | Ilexsaponin B2 | Ilexsaponin B2 is a saponin isolated from the root of Ilex pubescens Hook. |
| M42569 | Enpp-1-IN-16 | Enpp-1-IN-16 is an ENPP1 inhibitor. |
| M42568 | cis-Tadalafil | cis-Tadalafil is a PDE5 inhibitor (IC50: 0.09 μM). |
| M42567 | Motapizone | Motapizone (NAT 05-239) is a selective PDE3 inhibitor. |
| M42566 | PDE4-IN-13 | PDE4-IN-13 is a PDE4 inhibitor with an IC50 of 1.56 μM. |
| M42565 | PDE1-IN-5 | PDE1-IN-5 is a selective PDE1C inhibitor (IC50: 15 nM). |
| M42564 | CD00509 | CD00509 is a Tdp1 inhibitor, with an IC50 value of 0.71 μM. |
| M42563 | PDE5-IN-10 | PDE5-IN-10 is a potent PDE5 inhibitor with an IC50 of 20 nM. |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.
