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PDE Phosphodiesterase

Cat.No.  Name Information
M2030 Apremilast Apremilast is a novel, orally available small molecule inhibitor of PDE4 with IC50 of 74 nM.
M6804 IBMX IBMX is a pDE inhibitor (non-selective) with IC50 values of 6.5±1.2, 26.3±3.9 and 31.7±5.3 μM for PDE3, 4 and 5 respectively.
M9882 Roflumilast N-oxide Roflumilast N-oxide is a phosphodiesterase 4 inhibitor.
M9679 CP671305 CP671305 is a potent and selective, orally active inhibitor of phosphodiesterase-4-D with high activities.
M9347 ITI-214 phosphate ITI-214 phosphate is an orally active, potent and selective inhibitors of PDE1, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). ITI-214 inhibits recombinant full-length human PDE1A, PDE1B and PDE1C with Kis of 33 pM, 380 pM and 35 pM, respectively.
M8863 YM 976 Phosphodiesterase type IV (PDE4) inhibitor.
M8344 MBCQ MBCQ is selective inhibitor of cGMP-specific phosphodiesterase PDE V; IC50=19 nM.
M7429 Trequinsin hydrochloride Trequinsin hydrochloride is a extremely potent inhibitor of PDE3.
M6604 Cilostamide Cilostamide is a pDE3 inhibitor.
M6560 Carbazeran citrate Carbazeran citrate is a aldehyde oxidase substrate; PDE inhibitor.
M6287 GLPG1690 GLPG1690 (Ziritaxestat) is a first-in-class autotaxin (ATX) inhibitor, with IC50 of 131 nM and Ki of 15 nM.
M6153 E6005 RVT-501 (E6005) is a selective phosphodiesterase 4 (PDE4PDE4) inhibitor with an IC50 of 2.8 nM.
M6048 Vardenafil HCl Vardenafil Hcl is a PDE5 inhibitor used for treating erectile dysfunction.
M6042 Udenafil Udenafil(DA8159) is a PDE5 inhibitor used in urology to treat erectile dysfunction.
M6007 Theophylline Theophylline is a methylated xanthine derivative; competitive nonselective phosphodiesterase inhibitor and nonselective adenosine receptor antagonist.
M5960 Sildenafil Mesylate Sildenafil Mesylate is a mesylate form of Sildenafil, an inhibitor of Phosphodiesterase 5.
M5959 Sildenafil Sildenafil is a Phosphodiesterase 5 Inhibitor with IC50 of 5.22 nM.
M5939 Rolipram A selective inhibitor of PDE4, Rolipram, inhibits immunopurified PDE4B and PDE4D activity with IC50 of 130 nM and 240 nM, respectively. It has anti-inflammatory activity. Rolipram also increased cAMP levels and activated PKA, which in turn increased proteasome activity and inhibited tau aggregation.
M5833 Olprinone Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.
M5174 Icariin Icariin is a flavonol glycoside. Icariin inhibited PDE5 and PDE4 activity with IC50 of 432 nM and 73.50 μM, respectively. Icariin is also a PPARα activator.
M5060 Propentofylline Adamantane derivatives, processes for their preparation and pharmaceutical composition containing them.
M4964 HA130 HA130 is a selective ATX (autotaxin) inhibitor with IC50 of 28 nM.




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