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Autotaxin modulator 1

Cat. No. M11451

All AbMole products are for research use only, cannot be used for human consumption.

Autotaxin modulator 1  Structure
Size Price Availability Quantity
5mg USD 150  USD150 In stock
10mg USD 250  USD250 In stock
25mg USD 500  USD500 In stock
50mg USD 750  USD750 In stock
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Quality Control & Documentation
Biological Activity

Autotaxin Modulator 1 is an Autotaxin (ATX) inhibitor of Autotaxin (ATX). Autotaxin Modulator 1 is expected to be used for demyelination caused by injury or disease, as well as for the study of proliferative diseases such as tumors.

Chemical Information
Molecular Weight 543.54
Formula C28H31F6NO3
CAS Number 1548743-69-6
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Wayne Ng, et al. Adv Exp Med Biol. Lysophospholipid Signalling and the Tumour Microenvironment

[2] Naruomi Jinno, et al. Cancer Sci. Autotaxin in ascites promotes peritoneal dissemination in pancreatic cancer

[3] Joel Linden, et al. Annu Rev Immunol. Purine Release, Metabolism, and Signaling in the Inflammatory Response

[4] Victoria A Blaho, et al. Trends Pharmacol Sci. Crystal' Clear? Lysophospholipid Receptor Structure Insights and Controversies

[5] Natalie A Wheeler, et al. ASN Neuro. HIV-1 Tat Inhibits Autotaxin Lysophospholipase D Activity and Modulates Oligodendrocyte Differentiation

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Keywords: Autotaxin modulator 1 supplier, PDE, inhibitors, activators

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