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 About 30 results found for searched term "PDE" (0.011 seconds)

Cat.No.  Name Information
M1728 GSK256066 GSK256066 is a selective phosphodiesterase 4 (PDE4)inhibitor with an IC50 of 3.2 pM. *The compound is unstable in solutions, freshly prepared is recommended
M1734 BAY-60-7550 BAY-60-7550 is a potent PDE2 inhibitor with IC50 values of 2.0 nM (bovine) and 4.7 nM (human).
M1871 Roflumilast Roflumilast (trade names Daxas, Daliresp) is a novel and selective, long-acting inhibitor of phosphodiesterase 4 (PDE-4).
M1906 Piclamilast Piclamilast (RP 73401) is a potent and selective inhibitor of phosphodiesterase (PDE) 4.
M2030 Apremilast Apremilast is a novel, orally available small molecule inhibitor of PDE4 with IC50 of 74 nM.
M2410 Avanafil Avanafil is a highly selective PDE5 inhibitor with IC50 of 5.2 nM, >121-fold selectivity over other PDEs.
M2764 Ibudilast Ibudilast is a potent PDE4 inhibitor for PDE4A with IC50 of 54 nM.
M3337 Milrinone Milrinone is a potent and selective phosphodiesterase 3 inhibitor with an IC50 of 0.42 μM for the inhibition of FIII PDE.
M3375 S-(+)-Rolipram S-(+)-Rolipram inhibits human monocyte cyclic AMP-specific PDE4 with IC50 of 0.75 μM, has anti-inflammatory and anti-depressant activity in the central nervous system, less potent than its R enantiomer.
M3394 Deltarasin Deltarasin is a novel small molecule which inhibits the KRAS-PDEδ interaction and thus impairing oncogenic KRAS signalling.
M3434 Pimobendan Pimobendan is a selective inhibitor of PDE3 with IC50 of 0.32 μM.
M3437 Cilomilast Cilomilast is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity.
M3447 PF-2545920 PF-2545920 is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM, with >1000-fold selectivity over the PDE.
M3473 Tadalafil Tadalafil is a PDE-5 inhibitor with IC50 of 1.8 nM.
M3566 Vardenafil hydrochloride Trihydrate Vardenafil hydrochloride Trihydrate is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.
M4851 TAK-063 TAK-063 is a highly potent, selective and orally active PDE10A inhibitor with IC50 of 0.30 nM.
M5174 Icariin Icariin is a flavonol glycoside. Icariin inhibited PDE5 and PDE4 activity with IC50 of 432 nM and 73.50 μM, respectively. Icariin is also a PPARα activator.
M5519 Cilostazol Cilostazol is a potent cyclic nucleotide phosphodiesterase type 3 (PDE3) inhibitor with IC50 of 0.2 μM and inhibitor of adenosine uptake.
M5833 Olprinone Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.
M5939 Rolipram A selective inhibitor of PDE4, Rolipram, inhibits immunopurified PDE4B and PDE4D activity with IC50 of 130 nM and 240 nM, respectively. It has anti-inflammatory activity. Rolipram also increased cAMP levels and activated PKA, which in turn increased proteasome activity and inhibited tau aggregation.
M6042 Udenafil Udenafil(DA8159) is a PDE5 inhibitor used in urology to treat erectile dysfunction.
M6048 Vardenafil HCl Vardenafil Hcl is a PDE5 inhibitor used for treating erectile dysfunction.
M6153 E6005 RVT-501 (E6005) is a selective phosphodiesterase 4 (PDE4PDE4) inhibitor with an IC50 of 2.8 nM.
M6493 BC 11-38 BC 11-38 is a selective PDE11 inhibitor.
M6533 BRL 50481 BRL 50481 is a selective PDE7 inhibitor.
M6560 Carbazeran citrate Carbazeran citrate is a aldehyde oxidase substrate; PDE inhibitor.
M6574 CDP 840 hydrochloride CDP 840 hydrochloride is a potent and selective PDE4 inhibitor.
M6581 CGH 2466 dihydrochloride CGH 2466 dihydrochloride is a a 1, A 2B and A 3 antagonist and inhibitor of p38 MAPK and PDE4.
M6604 Cilostamide Cilostamide is a pDE3 inhibitor.
M6701 Eggmanone Eggmanone is a potent and selective PDE4 inhibitor; suppresses hedgehog signaling.

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