| Cat.No. | Name | Information |
|---|---|---|
| M2206 | TH-302 (Evofosfamide) | TH-302 is a highly potent and selective hypoxia-activated procompound targeting hypoxic regions of solid tumors with IC50 of 19 nM. |
| M6098 | Baicalein | Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor, IC50 value of 3.12 mM. |
| M9325 | EGTA | EGTA is a specific calcium chelator with a Kd of 60.5 nM at physiological pH (7.4) and a high specificity for Ca2+ than for Mg2+.EGTA significantly inhibits the substrate adhesion capacity of inflammatory macrophages. |
| M9330 | Brij-35 | Brij-35 (Polidocanol) is a high HLB, ethoxylated, nonionic ether of lauryl alcohol with broad pH stability. |
| M6154 | 2-PMPA tetrasodium | 2-PMPA (PMPA tetrasodium salt) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM. |
| M2250 | Pamidronate disodium | Pamidronate disodium is a nitrogen containing bisphosphonate, used to prevent osteoporosis. |
| M9916 | DPPH | DPPH (2,2-Diphenyl-1-picrylhydrazyl) is a stable free radical that measures the free radical scavenging activity of antioxidants. |
| M9194 | Insulin (human) | Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets. |
| M3409 | Formestane | Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM. |
| M9331 | 10-Hydroxy-trans-2-decenoic acid | 10-hydroxy-2-decenoic acid (10-H2DA) is the principal lipid component in royal jelly which is the food for queen and larvae honeybees. |
| M8107 | PF-6274484 | PF-6274484 is an irreversible EGFR kinase inhibitor that covalently reacts with active-site cysteine residues in the ATP binding pocket. |
| M8103 | CP724714 | CP724714 is a potent and selective inhibitor of HER2/ErbB2 with an IC50 value of 10 nM. |
| M8102 | PF-06422913 | PF-06422913 is an orally active, potent and selective metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator. |
| M8101 | PF-06412154 hydrochloride | PF-06412154 hydrochloride is a glucagon receptor antagonist. |
| M8098 | PF-06767832 | PF-06767832 is a cell permeable, potent and selective M1 muscarinic acetylcholine receptor Positive Allosteric Modulator (PAM). |
| M8097 | WAY 170523 | WAY 170523 is a potent and selective inhibitor of matrix metalloprotease MMP-13 (Collagenase-3), expressed in the skeleton during embryonic development, and sometimes highly overexpressed in human carcinomas and in chondrocytes and synovial cells in rheumatoid arthritis and osteoarthritis. |
| M8096 | PF-04937319 | PF-04937319 is a glucokinase activator with an EC50 value of 174 nM. |
| M8094 | PF-06761281 | PF-06761281 is an inhibitor of the sodium-coupled citrate transporter (NaCT or SLC13A5), which may be a target for tretment and prevention of metabolic disorders. |
| M8089 | PF-06747775 | PF-06747775 is an orally available, potent and selective inhibitor of the epidermal growth factor receptor) mutant form T790M (EGFR T790M inhibitor). |
| M8088 | PF-06284674 | PF-06284674 is a cell permeable, potent and selective M2 isoform of pyruvate kinase (PKM2) activator. |
| M8087 | PF-06459988 | PF-06459988 is an orally available irreversible inhibitor of epidermal growth factor receptor (EGFR) mutant (EGFRm) forms including the secondary acquired resistance mutation T790M. |
| M8086 | GRN-529 | GRN-529 is a brain penetrant, potent and selective negative allosteric modulator of the mGluR5 receptor (metabotropic glutamate receptor subtype 5) with an IC50 of 3. |
| M8085 | PF-06651481-00 | PF-06651481-00 is an isomer of orally available dual Src/Abl kinase inhibitor Bosutinib. |
| M8084 | PF-04753299 | PF-04753299 is a potent and selective inhibitor of LpxC (UDP-3-O-(R-3-hydroxymyri |
| M8082 | PF-05020182 | PF-05020182 is a Kv7. |
| M8081 | AG-17724 | AG-17724 is a potent peptidyl-prolyl isomerase (PPIase) Pin1 inhibitor. |
| M8079 | PF-3774076 | PF-3774076 is a CNS penetrant, potent, selective, partial agonist at the human α1A adrenoceptor. |
| M8078 | PF-06663195 | PF-06663195 is a potent inhibitor of β-site amyloid precursor protein (APP) Cleaving Enzyme 1 (BACE1, β-Secretase 1). |
| M8077 | PF-06649283 | PF-06649283 is a new β-Secretase (BACE) inhibitor. |
| M8076 | CP-101606 mesylate | CP-101606 mesylate (Traxoprodil mesylate) is a potent noncompetitive antagonist of N-methyl-D-aspartate (NMDA) receptors, selective for the NR2B subunit. |
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