GluR Glutamate receptor

Cat.No.	Name	Information
M2767	Ifenprodil Tartrate	Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM.
M9566	Glycine	Glycine is an inhibitory neurotransmitter in the CNS and also acts as a co-agonist along with glutamate.
M2884	NMDA	NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor.
M3003	CB-839	Telaglenastat (CB-839) is a potent, selective, and orally bioavailable glutaminase inhibitor with IC50 of 24 nM for recombinant human GAC.
M44821	Crocetin meglumine	Crocetin (Transcrocetin) meglumine, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity.
M42207	MPX-004	MPX-004 is a potent GluN2A antagonist.
M42206	GluN2B-NMDAR antagonist-1	GluN2B-NMDAR antagonist-1 is an orally active GluN2B-NMDAR antagonist.
M42205	Risevistinel	Risevistinel (NYX-783) is a positive allosteric modulator of N-methyl-D-aspartate (NMDA) receptor.
M42204	NMDA receptor antagonist 6	NMDA receptor antagonist 6 is an antagonist of NMDA receptor, targeting to the glycine binding site.
M42203	CP-465022	CP-465022 is a potent, and selective noncompetitive AMPA receptor antagonist with anticonvulsant activity.
M42202	Nevadistinel	Nevadistinel (NYX-458; NYX-3054) is a positive allosteric modulator of N-methyl-D-aspartate (NMDA) receptor.
M42201	NMDA receptor antagonist 7	NMDA receptor antagonist 7 is GluN2B subunit-selective NMDA Receptor antagonist, with an Ki of 93 nM and an IC50 of 72 nM.
M42200	NMDA receptor antagonist 8	NMDA receptor antagonist 8 is GluN2B subunit-selective NMDA Receptor antagonist, with an Ki of 265 nM and an IC50 of 62 nM.
M42199	DQP-26	DQP-26 is a potent NMDAR negative allosteric modulator with IC50 values of 0.77 μM and 0.44 μM for GluN2C and GluN2D, respectively.
M42198	UBP301 hydrochloride	UBP301 hydrochloride is a potent and selective antagonist of kainate receptor with IC50 and KD of 164 μM and 5.94 μM, respectively.
M42197	AMPA receptor modulator-4	AMPA receptor modulator-4, a 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide (BTD), is an orally active positive allosteric modulator of the AMPA receptors (AMPAR PAMs).
M41877	Z-Cyclopentyl-AP4	Z-Cyclopentyl-AP4 is a kainate-type glutamate receptor agonist (orthosteric agonist).
M41876	CVN636	CVN636 is a potent, orally active and selective mGluR7 allosteric agonist with an EC50 value of 7 nM for hu mGluR7.
M41875	mGluR3 modulator-1	mGluR3 modulator-1 is a mGluR3 modulator, with an EC50 of 1-10 μM in HEK293T-mGluR-Gqi5 Calcium Mobilization Assay.
M41874	LY456236	LY456236 is a selective, non-competitive and orally active mGlu1 receptor antagonist that inhibits phosphoinositide hydrolysis with an IC50 of 0.145 μM.
M41873	MK-8768	MK-8768 is a highly potent, orally bioavailable and selective class of mGluR2 negative allosteric modulator (IC50 of 9 .6nM) with excellent brain permeability.
M41872	Eglumegad hydrochloride	Eglumegad (LY354740) hydrochloride is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively.
M41871	IEM-1925 bromide	IEM-1925 bromide is an orally active glutamate receptor antagonist, increases the latent period and decreases the duration of status epilepticus in rats in a lithium-pilocarpine model of epilepsy.
M31234	Metapramine	Metapramine (19560 RP) is an antidepressant agent, inhibits norepinephrine reuptake, without affecting the reuptake of serotonin or dopamine. Metapramine is a low-affinity antagonist of the N-methyl-D-aspartic acid (NMDA) receptor complex channel.

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GluR Glutamate receptor

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