| Cat.No. | Name | Information |
|---|---|---|
| M2767 | Ifenprodil Tartrate | Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM. |
| M9566 | Glycine | Glycine is an inhibitory neurotransmitter in the CNS and also acts as a co-agonist along with glutamate. |
| M2884 | NMDA | NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. |
| M3003 | CB-839 | Telaglenastat (CB-839) is a potent, selective, and orally bioavailable glutaminase inhibitor with IC50 of 24 nM for recombinant human GAC. |
| M1897 | AZD6765 | AZD6765 is an NMDA receptor antagonist. |
| M58541 | VU0650786 | VU0650786 is a potent and selective CNS penetrant negative allosteric modulator of metabotropic glutamate receptor subtype 3 (mGlu3 NAM), with an IC50 of 392 nM. |
| M58534 | NS-102 | NS-102 is a selective kainate (GluK2) receptor antagonist. |
| M56817 | VU0424465 | VU0424465 is a potent and partial PAM (positive allosteric modulator)-agonist for mGlu5 mediated iCa2+ mobilization. |
| M56515 | ATPA | ATPA is a selective glutamate receptor GluR5 activator with EC50s of 0.66, 9.5, 1.4, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S741M), GluR5(S721T), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V), respectively. |
| M56514 | (R)-CPP | (R)-CPP is a highly potent NMDA receptor antagonist. |
| M56513 | UBP296 | UBP296 is a potent and selective antagonist of GLUK5-containing kainate receptor in the spinal cord. |
| M56512 | cis-ACPD | cis-ACPD is a potent agonist of NMDA receptor, with an IC50 of 3.3 μM. |
| M56511 | GNE-9278 | GNE-9278 is a highly selective positive allosteric modulator of NMDAR that acts at the GluN1 transmembrane domain (TMD). |
| M56510 | GYKI-47261 | GYKI-47261 is a competitive, orally active, and selective AMPA receptor antagonist with an IC50 of 2.5 μM. |
| M56509 | Rislenemdaz | Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC 50 of 8.1 nM and 3.6 nM, respectively. |
| M56508 | SDZ 220-581 | SDZ 220-581 is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. |
| M56507 | Neboglamine | Neboglamine (CR-2249; XY-2401) is a modulator for N-methyl-D-aspartate (NMDA) receptor. |
| M56506 | DL-AP5 sodium | DL-AP5 (2-APV) sodium is a competitive NMDA (N-methyl-D-aspartate) receptor antagonist. |
| M56505 | (R)-(+)-HA-966 | (R)-(+)-HA-966 ((+)-HA-966) is a partial agonist/antagonist of glycine site of the N-methyl-D-aspartate (NMDA) receptor complex. |
| M56504 | (S)-(-)-HA 966 | (S)-(-)-HA 966 ((-)-HA 966), a γ-Hydroxybutyrate-like agent, is weakly active as an NMDA-receptor antagonist. |
| M56503 | (2R,3S)-Chlorpheg | (2R,3R)-Chlorpheg is a week antagonist of L-homocysteic acid (L-HCA) induced depolarization.(2R,3R)-Chlorpheg also is a weak N-methyl-D-aspartate (NMDA) antagonist. |
| M56502 | 5-Iodowillardiine | 5-Iodowillardiine is a potent and selective kainate receptor agonist. |
| M56501 | NPEC-caged-(S)-AMPA | NPEC- caged-(S)-AMPA, a caged neurotransmitter analog, is a NPEC photoprotecting group caged the (S)-AMPA to make caged ligands specific for glutamate receptor sub-types. |
| M56500 | NMDAR antagonist 1 | NMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective NMDAR antagonist. |
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