| Cat.No. | Name | Information |
|---|---|---|
| M2767 | Ifenprodil Tartrate | Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM. |
| M9566 | Glycine | Glycine is an inhibitory neurotransmitter in the CNS and also acts as a co-agonist along with glutamate. |
| M2884 | NMDA | NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. |
| M3003 | CB-839 | CB-839 is a potent, selective, and orally bioavailable glutaminase inhibitor with IC50 of 24 nM for recombinant human GAC. |
| M6247 | VU6005649 | VU6005649 is a CNS penetrant mGlu7/8 receptor agonist with EC50s of 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively. |
| M6071 | Lu AF21934 | Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. |
| M5837 | Orphenadrine Citrate | Orphenadrine Citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects. |
| M5769 | Mephenesin | Mephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. |
| M5216 | SYM2206 | SYM2206 is a glutamate receptor antagonist with IC50 value of 2.8 μM. |
| M5157 | Perampanel | Perampanel is a selective noncompetitive AMPA-type glutamate receptor antagonist. |
| M5081 | CFM-2 | CFM-2 is a selective non-competitive AMPAR antagonist. |
| M5078 | (S)-Willardiine | (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. |
| M5076 | ZK200775 hydrate | ZK200775 hydrate is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. |
| M5071 | ZK200775 | ZK200775 is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. |
| M4957 | CIQ | CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. |
| M4956 | L-701324 | L-701324 is a long-acting oral anticonvulsant compound with high affinity and selectivity for glycine sites on NMDA receptors. |
| M4950 | Topiramate | Topiramate is an anticonvulsant that antagonizes GluR5 receptors and acts as a positive allosteric modulator of GABA receptor-mediated currents. |
| M4833 | Eliprodil | Eliprodil is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). |
| M3904 | Pulchinenoside A | Pulchinenoside can inhibit abnormal proliferation of synovial membrane by modulating Wnt pathway of RA rats.Pulchinenoside may inhibit the FLS proliferation in AA rats by increase in FLS apoptosis. |
| M3806 | GLYX-13 | GLYX-13 is a selective weak partial agonist of the glycine site of the NMDA receptor. |
| M3445 | ADX-47273 | ADX47273 is a potent and specific mGlu5 positive allosteric modulator(PAM) with EC50 of 0.17 μM, showing no activity at other mGlu subtypes. |
| M3279 | GYKI-52466 | GYKI-52466 is a non-competitive AMPA/kainate antagonists with IC50 of 7.5 μM and 11 μM, respectively. |
| M3189 | TCN-201 | TCN 201 is a NMDA receptor antagonist for NR1/NR2A and NR1/NR2B with pIC50 of 6.8 and 4.3, respectively. |
| M3126 | VU 0357121 | VU0357121 is a novel positive allosteric modulator (PAM) of mGlu5 with EC50 of 33 nM, is inactive or very weakly antagonizing at other mGlu receptor subtypes. |
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