Cat.No. | Name | Information |
---|---|---|
M2767 | Ifenprodil Tartrate | Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM. |
M9566 | Glycine | Glycine is an inhibitory neurotransmitter in the CNS and also acts as a co-agonist along with glutamate. |
M2884 | NMDA | NMDA(N-Methyl-D-aspartic acid)is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. |
M3003 | CB-839 | Telaglenastat (CB-839) is a potent, selective, and orally bioavailable glutaminase inhibitor with IC50 of 24 nM for recombinant human GAC. |
M7111 | PEPA | PEPA is a allosteric potentiator of AMPA receptor desensitization. |
M6846 | JNJ 16259685 | JNJ16259685 is a selective antagonist of mGlu1 receptor, and inhibits the synaptic activation of mGlu1 in a concentration-dependent manner with IC50 of 19 nM. |
M6691 | D-Serine | D-Serine is a potentiator, acts at glycine site. |
M6632 | CPPG | CPPG is a potent group III mGlu antagonist. |
M6619 | CNQX | CNQX (FG9065) is a potent and competitive AMPA/kainate receptor antagonist with IC50s of 0.3 μM and 1.5 μM, respectively. CNQX is a competitive non-NMDA receptor antagonist. |
M6438 | AMN 082 dihydrochloride | AMN 082 dihydrochloride is a the first selective mGlu 7 agonist. |
M6355 | 7-Chlorokynurenic acid sodium salt | 7-Chlorokynurenic acid sodium salt is a potent competitive inhibitor of L-glutamate uptake. Sodium salt of 7-Chlorokynurenic acid. |
M6338 | 3-MATIDA | 3-MATIDA is a potent, selective mGlu 1 antagonist. |
M6321 | 1-BCP | 1-BCP (Piperonylic acid piperidide) is a modulates AMPA-mediated responses. |
M6247 | VU6005649 | VU6005649 is a CNS penetrant mGlu7/8 receptor agonist with EC50s of 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively. |
M6071 | Lu AF21934 | Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. |
M5837 | Orphenadrine Citrate | Orphenadrine Citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects. |
M5769 | Mephenesin | Mephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. |
M5216 | SYM2206 | SYM2206 is a glutamate receptor antagonist with IC50 value of 2.8 μM. |
M5157 | Perampanel | Perampanel is a selective noncompetitive AMPA-type glutamate receptor antagonist. |
M5081 | CFM-2 | CFM-2 is a selective non-competitive AMPAR antagonist. |
M5078 | (S)-Willardiine | (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. |
M5076 | ZK200775 hydrate | ZK200775 hydrate is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. |
M5071 | ZK200775 | ZK200775 is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. |
M4957 | CIQ | CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. |
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