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MK-8768

Cat. No. M41873

All AbMole products are for research use only, cannot be used for human consumption.

MK-8768 Structure

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Quality Control & Documentation
Biological Activity

MK-8768 is a highly potent, orally bioavailable and selective class of mGluR2 negative allosteric modulator (IC50 of 9 .6nM) with excellent brain permeability.

Chemical Information
Molecular Weight 433.43
Formula C21H22F3N5O2
CAS Number 1432729-22-0
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Michael T Rudd et al. ACS Med Chem Lett. Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator

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  Catalog
Abmole Inhibitor Catalog




Keywords: MK-8768 supplier, GluR, inhibitors, activators

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