About 14 results found for searched term "GluR" (0.064 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2542 | CTEP | GluR |
| mGluR5 inhibitor | ||
| CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors. | ||
| M2724 | Gliquidone | Potassium Channel |
| Glurenorm | ||
| Gliquidone is an ATP-sensitive K+ channel antagonist with IC50 of 27.2 nM. | ||
| M9646 | Decoglurant | GluR |
| RG-1578; RO4995819 | ||
| Decoglurant (also known as RO4995819) is a negative allosteric modulator of the mGlu2 and mGlu3 receptors. | ||
| M14017 | Mavoglurant | GluR |
| AFQ056 | ||
| Mavoglurant (AFQ056) is a potent, selective, non-competitive and orally active mGluR5 antagonist, with an IC50 of 30 nM. | ||
| M14018 | Basimglurant | GluR |
| RG7090; CTEP Derivative | ||
| Basimglurant (RG7090) is a potent, selective and orally available mGlu5 negative allosteric modulator with a Kd of 1.1 nM. | ||
| M21797 | Auglurant | Others |
| Auglurant | ||
| M22211 | Dipraglurant | Others |
| ADX48621 | ||
| Dipraglurant | ||
| M22344 | Foliglurax monohydrochloride | Others |
| Foliglurax monohydrochloride | ||
| M27989 | Linaprazan glurate | Others |
| X842 | ||
| Linaprazan glurate inhibits exogenously or endogenously stimulated gastric acid secretion. Linaprazan glurate exhibits several advantageous properties, such as fast onset, high in vivo potency and/or long duration of action. Linaprazan glurate is useful in the research of gastrointestinal inflammatory diseases and peptic ulcer diseases. | ||
| M29073 | Valiglurax | GluR |
| VU0652957; VU2957 | ||
| Valiglurax (VU0652957) is a potent, orally active and selective mGlu4 positive allosteric modulator with EC50 values of 64.6 nM and 197 nM for hmGlu4/Gqi5 and rmGlu4 GIRK, respectively. Valiglurax is a central nervous system (CNS) penetrant. Valiglurax can be used in research of Parkinson's disease. | ||
| M41188 | TAT-GluR23A Fusion Peptide | Anti-infection |
| TAT-GluR23A Fusion Peptide is a biological active peptide. | ||
| M41875 | mGluR3 modulator-1 | GluR |
| mGluR3 modulator-1 is a mGluR3 modulator, with an EC50 of 1-10 μM in HEK293T-mGluR-Gqi5 Calcium Mobilization Assay. | ||
| M43344 | GluR23Y | Others |
| GluR23Y is a biological active peptide. | ||
| M51827 | Tat-GluR23Y, scrambled | Amino Acid Derivatives |
| Tat-GluR23Y, scrambled is the scrambled peptide of Tat-GluR23Y. | ||
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