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Decoglurant

Cat. No. M9646

All AbMole products are for research use only, cannot be used for human consumption.

Decoglurant Structure
Synonym:

RG-1578; RO4995819

Size Price Availability Quantity
5mg USD 248  USD248 In stock
10mg USD 365  USD365 In stock
25mg USD 655  USD655 In stock
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Quality Control & Documentation
Biological Activity

Decoglurant (also known as RO4995819) is a negative allosteric modulator of the mGlu2 and mGlu3 receptors.

Chemical Information
Molecular Weight 447.34
Formula C21H11F6N5
CAS Number 911115-16-7
Solubility (25°C) DMSO ≥ 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Samuel T Wilkinson, et al. Drv g Discov Today. A new generation of antidepressants: an update on the pharmaceutical pipeline for novel and rapid-acting therapeutics in mood disorders based on glutamate/GABA neurotransmitter systems

[2] H Javelot. Ann Pharm Fr. Psychopharmacology of anxiety and depression: Historical aspects, current treatments and perspectives

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Keywords: Decoglurant, RG-1578; RO4995819 supplier, GluR, inhibitors, activators

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