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Gliquidone

Cat. No. M2724

All AbMole products are for research use only, cannot be used for human consumption.

Gliquidone Structure
Synonym:

Glurenorm

Size Price Availability Quantity
50mg USD 55  USD55 In stock
100mg USD 65  USD65 In stock
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Quality Control & Documentation
Biological Activity

Gliquidone is an ATP-sensitive K+ channel antagonist with IC50 of 27.2 nM.

Chemical Information
Molecular Weight 527.63
Formula C27H33N3O6S
CAS Number 33342-05-1
Solubility (25°C) DMSO 85 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jieun Kim, et al. The Anti-diabetic Drug Gliquidone Modulates Lipopolysaccharide-Mediated Microglial Neuroinflammatory Responses by Inhibiting the NLRP3 Inflammasome

[2] Rui Zhang, et al. Gliquidone ameliorates hepatic insulin resistance in streptozotocin-induced diabetic Sur1 -/- rats

[3] Hengyu Tian, et al. Gliquidone Alleviates Diabetic Nephropathy by Inhibiting Notch/Snail Signaling Pathway

[4] Thomas Gelbrich, et al. Gliquidone

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Keywords: Gliquidone, Glurenorm supplier, Potassium Channel, inhibitors, activators

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