| Cat.No. | Name | Information |
|---|---|---|
| M3754 | Nedocromil | Nedocromil is a pyranoquinolone derivative that inhibits activation of inflammatory cells which are associated with asthma, including eosinophils, neutrophils, macrophages, mast cells, monocytes, and platelets. |
| M3665 | Promethazine hydrochloride | Promethazine hydrochloride is a potent histamine H1 receptor antagonist used as a sedative and antiallergic compound. |
| M3487 | Azelastine hydrochloride | Azelastine hydrochloride is a potent, second-generation, selective, histamine antagonist. |
| M3458 | Chlorpheniramine Maleate | Chlorpheniramine (Chlorpheniramine maleate, Chlorphenamine) is an histamine H1 receptor antagonist with IC50 of 12 nM. |
| M3454 | Olopatadine hydrochloride | Olopatadine hydrochloride is a histamine blocker and mast cell stabilizer with an IC50 of 559 μM for the release of histamine. It can be used in studies related to allergic conjunctivitis and rhinitis. |
| M3431 | Nizatidine | Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM. |
| M3385 | Cimetidine | Cimetidine, a histamine congener, competitively inhibits histamine binding to histamine H2 receptors. |
| M3383 | Diphenhydramine hydrochloride | Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB). |
| M3318 | Clemastine Fumarate | Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM. |
| M3226 | Brompheniramine hydrogen maleate | Brompheniramine hydrogen maleate is a histamine H1 receptors antagonist. |
| M3213 | Meclizine dihydrochloride | Meclizine is a histamine H1 receptor antagonist used to treat nausea and motion sickness, has anti-histamine, anti-muscarinic and anti-oxidative phosphorylation properties, also an agonist ligand for mCAR (constitutive androstane receptor) and an inverse agonist for hCAR. Phase2. |
| M3091 | Tripelennamine hydrochloride | Tripelennamine is a widely used H1 antagonist, inhibiting PhIP glucuronidation with IC50 of 30 μM. |
| M2990 | Rupatadine Fumarate | Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively. |
| M2971 | Pyrilamine Maleate | Pyrilamine is a histamine H1 receptor inverse agonist, it binds to a G protein-coupled form of the receptor and promotes a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11-mediated signaling. |
| M2935 | Pheniramine Maleate | Pheniramine Maleate is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria. |
| M2919 | Pemirolast potassium | Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent. |
| M2811 | Levodropropizine | Levodropropizine possess anti-allergic and inhibits histamine receptor, reduces cough by interfering with stimulus activation of peripheral endings of sensory nerves and by modulation of neuropeptides involved in the cough reflex. |
| M2784 | JNJ-7777120 | JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM, exhibits >1000-fold selectivity over the other histamin receptors. |
| M2760 | Hydroxyzine dihydrochloride | Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM. |
| M2756 | Histamine dihydrochloride | Histamine 2HCl is an endogenous ligand for the histamine receptor, which can cause allergic reactions by interacting with H1 receptors, promote acid secretion by interacting with H2 receptors, as well as inhibit histamine release and modulate immune responses by interacting with H3 receptors and H4 receptors. It can be used in studies related to allergy, hyperacidity, sleep disorders, asthma and many other diseases. |
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