| Cat.No. | Name | Information |
|---|---|---|
| M56361 | Dimethindene | Dimethindene is a potent, selective histamine H1 antagonist. |
| M56228 | ABT-288 | ABT-288 is a competitive, potent and selective histamine H3 receptor (H3R) antagonist. |
| M56227 | A-349821 | A-349821 is a histamine H3 receptor antagonist characterized as a radioligand ([3H]-A-349821) for in vivo receptor occupancy assessment. |
| M56226 | Betazole | Betazole (Ametazole), a pyrazole analogue of histamine, is an orally active histamine H2 receptor agonist. |
| M56225 | Tiotidine | Tiotidine (ICI 125211) is a potent and selective antagonist of histamine H2-receptor (pA2=7.3-7.8 for guinea-pig right atrium). |
| M56224 | Amthamine | Amthamine is a histamine receptor (H1R-H4R) agonist. |
| M56223 | Enerisant | Enerisant (TS-091) is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively. |
| M56222 | Lodoxamide | Lodoxamide (U-42585E free acid) is an antiallergic compound acting as a mast-cell stabilizer for the treatment of asthma and allergic conjunctivitis. |
| M56221 | PF-03654764 | PF-03654764 is an orally active, selective histamine H3 receptor antagonist with Ki values of 1.2 nM and 7.9 nM for human H3 and rat H3 in whole cell assay, respectively. |
| M56220 | Alimemazine | Alimemazine is an antipruritic agent and also a hemagglutinin (HA)-receptor antagonist.Alimemazine (Trimeprazine) is also acts as a partial agonist against the histamine H1 receptor (H1R) and other GPCRs. |
| M56219 | Niperotidine | Niperotidine is a histamine H2-receptor antagonist. |
| M56218 | Thioperamide | Thioperamide (MR-12842) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. |
| M56217 | ROS 234 dioxalate | ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. |
| M56216 | Dexchlorpheniramine | Dexchlorpheniramine is an potent and blood-brain barrier (BBB) penetrant histamine 1 (H1) receptor antagonist with anticholinergic properties. |
| M56215 | (±)-Carbinoxamine | (±)-Carbinoxamine is a histamine H1 receptor antagonist. |
| M56214 | Enerisant hydrochloride | Enerisant (TS-091) hydrochloride is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively. |
| M56213 | Alimemazine hemitartrate | Alimemazine hemitartrate is a phenothiazine derivative that is generally used as an antipruritic agent and also a hemagglutinin (HA)-receptor antagonist. |
| M56212 | Betazole dihydrochloride | Betazole (Ametazole) dihydrochloride, a pyrazole analogue of histamine, is an orally active H2 receptor agonist. |
| M56211 | Betahistine EP Impurity C | Betahistine EP Impurity C (NSC19005) is an impurity of Betahistine. |
| M56210 | Immethridine dihydrobromide | Immethridine dihydrobromide is a selective histamine H3 receptor (H3R) agonist. |
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