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Histamine Receptor Histamine Receptor

Cat.No.  Name Information
M2755 Histamine Phosphate Histamine Phosphate is an endogenous ligand for the histamine receptor that can induce allergic reactions by acting with H1 receptors, promote acid secretion by acting with H2 receptors, and inhibit histamine release and modulate immune responses by acting with H3 receptors and H4 receptors. It can be used in studies related to allergy, hyperacidity, sleep disorders, asthma and many other diseases.
M2699 Fexofenadine hydrochloride Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
M2697 Fenspiride hydrochloride Fenspiride hydrochloride is a bronchodilator with anti-inflammatory properties, inhibiting phosphodiesterase 4 and phosphodiesterase 3 activities with logIC50 values of 4.16 and 3.44, respectively, in human isolated bronchi.
M2671 Epinastine hydrochloride Epinastine hydrochloride is an antihistamine and mast cell stabilizer. Epinastine hydrochloride is a potent, selective and orally-active histamine H1 receptor antagonist.
M2660 Ebastine Ebastinea is an orally active, potent histamine H1 receptor antagonist for studies related to allergic diseases.
M2653 Doxylamine Succinate Doxylamine succinate competitively inhibits histamine at H1 receptors with substantial sedative and anticholinergic effects.
M2650 Doxepin hydrochloride Doxepin hydrochloride is a potent and selective histamine receptor H1 antagonist. Doxepin hydrochloride is also a potent CYP450 inhibitor and significantly inhibits CYP450 2C19 and 1A2.
M2643 Diphenylpyraline hydrochloride Diphenylpyraline hydrochloride (DPP) is an internationally available antihistamine that produces therapeutic antiallergic effects by binding to histamine H₁ receptors.
M2639 Dimaprit dihydrochloride Dimaprit is a histamine type 2 receptor agonist.
M2621 Desloratadine Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
M2582 Clemizole Clemizole is a H1 histamine receptor antagonist with IC50 Value of 8 mM (NS4B).
M2545 Cyclizine dihydrochloride Cyclizine 2HCl is a piperazine derivative with Histamine H1 receptor antagonist activity.
M2522 Ciproxifan Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
M2477 Buclizine hydrochloride Buclizine hydrochloride is an antihistamine and anticholinergic of the piperazine derivative family.
M2452 Betahistine dihydrochloride Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.
M2449 Bepotastine Besilate Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
M2416 Azatadine dimaleate Azatadine dimaleate is an antihistamine and anticholinergic compound with IC50 of 6.5nM and 10nM, respectively.
M2413 Azacyclonol Azacyclonol, also known as γ-pipradol, which diminishes hallucinations in psychotic individuals.
M2398 Antazoline hydrochloride Antazoline hydrochloride is a first generation antihistamine, binding to the histamine H1 receptor and blocking the action of endogenous histamine.
M2088 Ciproxifan maleate Ciproxifan is an orally bioavailable, extremely potent histamine H3 inverse agonist/antagonist.




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