| Cat.No. | Name | Information |
|---|---|---|
| M20574 | Thonzylamine | Thonzylamine is an antihistamine and anticholinergic drug. |
| M20520 | Chloropyramine hydrochloride | Chloropyramine hydrochloride is a histamine receptor H1 antagonist and has anti-cholinergic, antispasmodic, and antiallergic effects. |
| M20515 | Emedastine | Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM). |
| M20511 | Betahistine | Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug. |
| M20495 | Cloperastine hydrochloride | Cloperastine is a drug with a central antitussive effect, and is also endowed with an antihistaminic activity. |
| M20424 | CarbinoxaMine Maleate | Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties. |
| M13995 | Adriforant hydrochloride | Adriforant hydrochloride (PF-3893787 hydrochloride) is a novel histamine H4 receptor antagonist binding affinity (Ki=2.4 nM) and is also a functional (Ki=1.56 nM) antagonist. |
| M13994 | N-Acetylhistamine | N-Acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions. |
| M13992 | Chlorcyclizine hydrochloride | Chlorcyclizine hydrochloride is a histamine H1 antagonist. |
| M13991 | Bepotastine | Bepotastine is a selective and orally active second-generation histamine H1 receptor antagonist. Bepotastine has the potential for allergic rhinitis, allergic conjunctivitis and urticaria/pruritus research. |
| M11287 | JNJ-39758979 | Jnj-39758979 is a selective, orally active, high-affinity histamine H4 receptor antagonist with Ki values of 12.5, 5.3 and 25 nM for human, mouse and monkey histamine H4 receptor, respectively. Jnj-39758979 antagonized histamine-induced cAMP inhibition with a pA2 of 7.9. Jnj-39758979 has good anti-inflammatory and antipruritic effects. |
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