| Cat.No. | Name | Information |
|---|---|---|
| M2489 | Carbachol chloride | Carbachol is a cholinomimetic compound that binds and activates the acetylcholine receptor. |
| M3470 | Oxybutynin | Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties. |
| M3190 | PNU-282987 | PNU-282987 is a highly selective α7 nAChR agonist with Ki of 27 nM. |
| M5683 | Glycopyrrolate | Glycopyrrolate(Glycopyrronium Br) is a muscarinic competitive antagonist used as an antispasmodic. |
| M42638 | hAChE/hBACE-1-IN-2 | hAChE/hBACE-1-IN-2 is a potent, orally active, blood-brain barrier transboundary triple inhibitor of hAChE, hBChE, and HACE-1 with IC50s of 0.113 μM, 1.48 μM and 0.38 μM, respectively. |
| M42637 | SB-1436 | SB-1436 is an Cholinesterase (ChE) inhibitor, inhibits AChE, BChE and rHuAChE with IC50s of 0.176, 0.37 and 0.08 μM, respectively. |
| M42214 | Tebanicline hydrochloride | Tebanicline hydrochloride (Ebanicline hydrochloride) is a nAChR modulator with potent, orally effective analgesic activity. |
| M42213 | CVN417 | CVN417 is an orally active α6 subunit-containing nAChR antagonist, modulating phasic dopaminergic neurotransmission in an impulse-dependent manner. |
| M42212 | Epiboxidine hydrochloride | Epiboxidine hydrochloride is a potent and selective neural nAChR agonist with Kis of 0.46 nM and 1.2 nM for rat and human α4β2 nAChRs, respectively. |
| M42211 | TC-1698 | TC-1698 is a selective α7 nicotinic acetylcholine receptors agonist with EC50 value of 0.16 μM and 0.46 μM for monkey α7 nicotinic receptor and human α7 nicotinic receptor, respectively. |
| M41867 | Oxyphenonium bromide | Oxyphenonium bromide is an antiacetylcholine compound. |
| M41866 | Nitrocaramiphen hydrochloride | Nitrocaramiphen hydrochloride is a selective M1 receptor antagonist (Ki: 5.5 nM). |
| M41865 | J-104129 | J-104129 is a selective and orally active muscarinic M3 receptor antagonist (Ki = 4.2 nM). |
| M41864 | Muscarine | Muscarine ((+)-Muscarine) is a toxin that can stimulate the parasympathetic nervous system. |
| M41863 | Milameline hydrochloride | Milameline (CI 979) hydrochloride is a muscarinic receptor agonist that improves cognition. |
| M41862 | Dipeptide diaminobutyroyl benzylamide diacetate | Dipeptide diaminobutyroyl benzylamide diacetate, a Wagerlin-1-mimicking peptide, is a mAChR antagonist. |
| M41861 | VU0364572 TFA | VU0364572 TFA is an orally active and selective allosteric agonist of the M1 muscarinic receptor with an EC50 of 0.11 μM. |
| M41860 | Arecaidine but-2-ynyl ester tosylate | Arecaidine but-2-ynyl ester tosylate (ABET) is a selective mAChR M2 agonist that dose-dependently decreases mean arterial pressure and heart rate in rats. |
| M41000 | (R)-Oxybutynin | (R)-Oxybutynin is a racemic isomer of Oxybutynin and an orally active muscarinic receptor antagonist. It has antitussive and anticholinergic activity, competitively antagonizes carbachol-induced contractions, and can be used in studies related to obstructive sleep apnea (OSA). |
| M40911 | Octahydroaminoacridine succinate | Octahydroaminoacridine succinate is a Tacrine analog and a potent inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). It may be used in studies related to Alzheimer's disease (AD). |
| M39202 | Cyclopenin | Cyclopenin ((±)-Isocyclopenine) is a racemate. |
| M39201 | Lycodoline | Lycodoline is a alkaloid with butyrylcholinesterase (BChE) (IC50 of 667 μM) inhibition activities. |
| M39200 | Vomifoliol | Vomifoliol, a compound related to abscisie acid (ABA), has a modified 2,4-pentadiene side chain and has activity equal to that displayed by ABA. Vomifoliol exhibits antiacetylcholinesterase activity and displays moderate antileishmanial activity. |
| M39199 | Isonaringin | Isonaringin shows anti-Alzheimer’s activity by inhibiting AChE. |
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