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CVN417

Cat. No. M42213

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CVN417 Structure

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Quality Control & Documentation
Biological Activity

CVN417 is an orally active α6 subunit-containing nAChR antagonist, modulating phasic dopaminergic neurotransmission in an impulse-dependent manner.

Chemical Information
Molecular Weight 362.85
Formula C18H23ClN4O2
CAS Number 2919851-73-1
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Cristiano Bolchi et al. J Med Chem. Addressing Motor Dysfunction by a Selective α6-Containing Nicotinic Receptor Antagonist

[2] Louisa A Christie et al. J Med Chem. Discovery of CVN417, a Novel Brain-Penetrant α6-Containing Nicotinic Receptor Antagonist for the Modulation of Motor Dysfunction

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Keywords: CVN417 supplier, AChR/AChE, inhibitors, activators

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