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Epiboxidine hydrochloride

Cat. No. M42212

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Epiboxidine hydrochloride Structure

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Quality Control & Documentation
Biological Activity

Epiboxidine hydrochloride is a potent and selective neural nAChR agonist with Kis of 0.46 nM and 1.2 nM for rat and human α4β2 nAChRs, respectively.

Chemical Information
Molecular Weight 214.69
Formula C10H15ClN2O
CAS Number 862909-67-9
Form Solid
Storage -20°C, dry, sealed
References

[1] Clelia Dallanoce et al. Chirality. The enantiomers of epiboxidine and of two related analogs: synthesis and estimation of their binding affinity at α4β2 and α7 neuronal nicotinic acetylcholine receptors

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