| Cat.No. | Name | Information |
|---|---|---|
| M19285 | Vitamin A | Vitamin A (Retinol) is a naturally occuring fat-soluble vitamin that is important for normal vision, the immune system, and reproduction. It also plays roles in normal functioning of heart, lungs, kidneys, and other organs. |
| M2241 | Adapalene | Adapalene is a third-generation topical retinoid, it is a potent RAR agonist, with AC50 values of 2.3 nM, 9.3 nM, and 22 nM for RARβ, RARγ, RARα, respectively. Adapalene also inhibits the enzymatic activity of GOT1 in a non-competitive manner. Adapalene is also an MST1 agonist. |
| M7568 | AM580 | AM580 is a selective RARα agonist with IC50 and EC50 of 8 nM and 0.36 nM, respectively. |
| M7568 | AM580 | AM580 is a selective RARα agonist with IC50 and EC50 of 8 nM and 0.36 nM, respectively. |
| M7097 | PA 452 | PA 452 is a rXR antagonist. |
| M6573 | CD 2665 | CD 2665 is a selective RARβ/γ antagonist. |
| M6521 | BMS 753 | BMS 753 is a rARα-selective agonist. |
| M6416 | AGN 193109 | AGN 193109 is a high affinity pan-RAR (retinoic acid receptors) antagonist, with Kds of 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ, respectively. |
| M6155 | AR7 | AR7 is a retinoic acid receptor α (RARα) antagonist, it specifically activates chaperone-mediated-autophagy (CMA) activity without affecting macroautophagy. |
| M5455 | Bexarotene | Bexarotene (LGD1069) is a retinoid specifically selective for retinoid X receptors, used as an oral antineoplastic agent in the treatment of cutaneous T-cell lymphoma. |
| M4774 | 11-hydroxy-sugiol | 11-hydroxy-sugiol |
| M3973 | Tazarotene | Tazarotene (AGN 190168) is a new member of the acetylenic class of RARβ/γ selective retinoids which is approved to treat a variety of skin diseases, exhibits an anti-proliferative effect in human basal cell carcinoma (BCC) by triggering caspase-dependent apoptosis. |
| M3150 | Fenretinide | Fenretinide (4-HPR) is a synthetic retinoid deriverative. Fenretinide is shown to exhibit binding to the retinoic acid receptors (RAR) at concentrations necessary to induce cell death. |
| M3094 | TTNPB | TTNPB (Arotinoid Acid) is a potent RAR agonist, and inhibits binding of [3H]tRA with IC50 of 5.1 nM, 4.5 nM, and 9.3 nM for human RARα, β, and γ, respectively. |
| M3049 | Tamibarotene | Tamibarotene is a synthetic retinoic acid receptor (RAR) agonist with high specificity for RARα and RARβ over RARγ. |
| M1961 | Acitretin (Ro 10-1670) | Acitretin (Ro 10-1670) is a second-generation retinoid. |
| M56789 | YCT529 | YCT529 is a potent, selective and orally active RAR-α inhibitor. |
| M56788 | LG101506 | LG101506 is a selective and orally active RXR modulator with a Ki of 2.7 nM for RXRα. |
| M56787 | ER 50891 | ER-50891 is a potent antagonist of retinoic acid receptor α(RARα). |
| M56786 | LG100754 | LG100754 (UVI 2112) is a RXR dimers modulater. |
| M56785 | AGN 196996 | AGN 196996 is a potent and selective RARα antagonist with Ki value of 2 nM; little binding affinity for RARβ(Ki=1087 nM) and RARγ(Ki=8523 nM). |
| M56784 | Ro 41-5253 | Ro 41-5253 is an orally active selective retinoic acid receptor alpha (RARα) antagonist. |
| M56783 | YCT529 free acid | YCT529 free acid is a potent, selective and orally active RAR-α inhibitor. |
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