| Cat.No. | Name | Information |
|---|---|---|
| M3326 | Memantine hydrochloride | Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively. |
| M2079 | Chrysin | Chrysin is a naturally occurring flavone chemically extracted from the passion flowers Passiflora caerulea. |
| M40620 | TP0472993 | TP0472993 is a novel, orally active, selective inhibitor of 20-hydroxyeicosatetraenoic acid (20-HETE) synthesis that inhibits the production of 20-HETE, thereby reducing the ERK1/2 and STAT3 signaling pathways, and ultimately inhibiting the progression of renal fibrosis. It can be used in studies related to chronic kidney disease (CKD). |
| M22269 | 1-Ethynylnaphthalene | 1-Ethynylnaphthalene |
| M21184 | Soticlestat | Soticlestat (TAK-935; OV935) is a first-in-class, potent, selective, orally active inhibitor of cholesterol 24-hydroxylase (CH24H), which is used in the study of epilepsy syndromes. |
| M21085 | Pregnenolone 16α-carbonitrile | Pregnenolone 16α-carbonitrile is a derivative of pregnendione that functions as an agonist of the rodent pregnane X receptor (PXR). pregnenolone 16α-carbonitrile is a synthetic steroid that induces expression of cytochrome P450 3A. Pregnenolone 16α-carbonitrile exhibits greater tolerance to subsequent stress injury. |
| M19949 | Phloracetophenone | Phloracetophenone, or 2,4,6-trihydroxyacetophenone (THA), the aglycone component of phloracetophenone glucoside, is a naturally occurring compound obtained from the rhizome of Curcuma comosa (Family Zingiberaceae). |
| M19353 | Fraxinol | Fraxinol is isolated from Lobelia chinensis. |
| M14311 | Cecropin B | Cecropin B has high level of antimicrobial activity and is considered as a valuable peptide antibiotic. |
| M14310 | Bergamottin | Bergamottin is a potent and competitive CYP1A1 inhibitor with a Ki of 10.703 nM. |
| M11528 | Naringin | Naringin, a flavanone glycoside, exerts various of pharmacological effects such as blood lipid lowering, antioxidant activity, anticancer activity, and inhibition of cytochrome P450 enzymes. |
| M11176 | Tebuconazole | Tebuconazole is an agricultural azole fungicide that also inhibits CYP51 for Candida albicans CYP51 (CaCYP51) and truncated human CYP51 (Δ60HsCYP51). IC50 The values are 0.9 and 1.3 μM, respectively. |
| M11164 | SDZ285428 | SDZ285428 is a CYP51 inhibitor. SDZ285428 suppresses Trypanosoma cruzi (TC) CYP51, I/E2 <1 (5 min) and I/E2=9 (1 h). SDZ285428 suppresses Trypanosoma brucei (TB) CYP51, I/E2 <1 (5 min) and I/E2=35 (1 h). |
| M11137 | Dihydromethysticin | Dihydroestherol (Dihydromethysticin) kava lactone, with induced CYP3A23 activity. |
| M10656 | Bergaptol | Bergaptol is a hydroxylated psoralen that acts as a potent inhibitors of debenzylation activity of CYP3A4 enzyme with an IC50 value of 24.92 uM. |
| M10488 | Phthalic acid mono-2-ethylhexyl ester (liquid) | Phthalic acid mono-2-ethylhexyl ester (MEHP) is a major bioactive metabolite of diethylhexyl phthalate (DEHP), which inhibits the 17, 20 lyase activity of CYP17. |
| M10057 | α-Naphthoflavone | α-Naphthoflavone is a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. |
| M9931 | ε-Viniferin | ε-Viniferin is a potent inhibitor for all the CYP family, with Ki values from 0.5-20 μM. |
| M9877 | Rhapontigenin | Rhapontigenin is a selective inactivator of cytochrome P450 1A1 with IC50 of 400 nM. |
| M9684 | (Rac)-Brassinazole | (Rac)-Brassinazole is a brassinosteroid (BR) biosynthesis inhibitor. |
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