| Cat.No. | Name | Information |
|---|---|---|
| M3326 | Memantine hydrochloride | Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively. |
| M2079 | Chrysin | Chrysin is a naturally occurring flavone chemically extracted from the passion flowers Passiflora caerulea. |
| M4000 | (±)-Naringenin | (±)-Naringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines. |
| M2929 | PF-4981517 | PF-4981517 is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM, exhibits >500-fold selectivity over CYP3A5 and CYP3A7. |
| M2537 | Cobicistat | Cobicistat (GS-9350) is a potent and selective inhibitor of CYP3A with IC50 of 30-285 nM. |
| M2515 | Chlorzoxazone | Chlorzoxazone is a probe for human liver cytochrome P-450IIE1. |
| M2058 | Ketoconazole | Ketoconazole (R-41400) is an imidazole anti-fungal agent, a CYP3A4 and CYP24A1 inhibitor. |
| M1833 | Imidaclopride | Imidaclopride is a systemic insecticide which acts as an insect neurotoxin and belongs to a class of chemicals called the neonicotinoids. |
| M1814 | Avasimibe | Avasimibe (CI-1011) is a novel orally bioavailable ACAT inhibitor with IC50 values of 2.9, 13.9, 26.5 µM for CYP2C9, CYP1A2 and CYP2C19, respectively. |
| M1636 | Abiraterone | Abiraterone acetate (CB-7598) is a potent, selective, and orally available inhibitor of CYP17 with an IC50 of 4 nM. |
| M56608 | MS-PPOH | MS-PPOH is a potent and selective cytochrome P450 (CYP) epoxygenase inhibitor. |
| M56607 | (R)-Mephenytoin | (R)-Mephenytoin ((-)-Mephenytoin), the R-enantiomer of Mephenytoin. |
| M56606 | (3S,5S)-Atorvastatin | (3S,5S)-Atorvastatin is a inactive enantiomer of Atorvastatin. |
| M56605 | (3S,5S)-Atorvastatin sodium salt | (3S,5S)-Atorvastatin sodium salt is a pregnane X receptor (PXR) activator and the inactive enantiomer of Atorvastatin. |
| M56604 | Fadrozole hydrochloride hemihydrate | Fadrozole hydrochloride hemihydrate is an orally active, potent, selective and nonsteroidal aromatase inhibitor, with an IC50 of 6.4 nM. |
| M52647 | Cytochrome P450 reductase | Cytochrome P450 reductase is a NADPH-cytochrome reductase. |
| M45355 | 20-SOLA | 20-SOLA is a water-soluble 20-HETE antagonist. |
| M45354 | TS-011 | TS-011 is a selective inhibitor of 20-hydroxyeicosatetraenoic acid (20-HETE) synthesis. |
| M45353 | Dibromo-dodecenyl-methylsulfimide | Dibromo-dodecenyl-methylsulfimide is a selective inhibitor of 20-HETE synthesis and attenuates the vasodilatory response to sodium nitroprusside (SNP). |
| M45022 | Terpinyl acetate | α-Terpinyl acetate is a monoterpene ester isolated from Laurus nobilis L. |
| M44872 | Harmidol hydrochloride | Harmalol hydrochloride, a beta carboline alkaloid, presents in several medicinal plants such as Peganum harmala. |
| M44743 | 4'-Methylchrysoeriol | 4'-Methylchrysoeriol is a potent inhibitor of Cytochrome P450 enzymes, with an IC50 of 19 nM for human P450 1B1-dependent EROD. |
| M44695 | 2',5,6',7-Tetrahydroxyflavone | 5,7,2',6'-Tetrahydroxyflavone is a natural flavonoid that inhibits hepatic testosterone 6β-hydroxylation (CYP3A4) activity with an IC50 of 7.8 μM. |
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