| Cat.No. | Name | Information |
|---|---|---|
| M7325 | Rimonabant Hydrochloride | Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity |
| M8919 | BAY 59-3074 | BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively. |
| M7613 | 2-Arachidonyl glycerol | 2-Arachidonyl glycerol is an endogenous cannabinoid and also an agonist at cannabinoid receptors. |
| M6778 | GW 405833 | GW 405833 is a selective, high affinity CB2 receptor partial agonist. |
| M6429 | AM 630 | AM 630 is a CB2 selective inverse agonist. |
| M6402 | ACPA | ACPA is a potent, selective CB 1 agonist. |
| M5290 | (±)-SLV-319 | (±)-SLV319 (Ibipinabant) is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo. |
| M4777 | Pregnenolone | Pregnenolone (3β -hydroxy-5-pregnen-20-one) is a powerful neurosteroid, and is the major precursor of various steroids, including steroids. Pregnenolone is a specific signaling inhibitor of cannabinoid CB1 receptor. |
| M3282 | GW842166X | GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. |
| M3266 | WIN 55212-2 mesylate | WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively. |
| M2981 | Rimonabant | Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane. |
| M2552 | Otenabant | Otenabant (CP-945598) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM. |
| M2461 | BML-190 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| M2379 | AM251 | AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain. |
| M2343 | AM-2201 | AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively. |
| M2051 | CP 945598 hydrochloride | CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively). |
| M2012 | AM1241 | AM1241 is a cannabinoid CB2 receptor selective agonist. |
| M1907 | Org 27569 | Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor. |
| M56153 | UCM707 | UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of Anandamide. |
| M56152 | SCH 336 | SCH 336 is a potent, selective, inverse and orally active CB2 agonist. |
| M56151 | JTE-907 | JTE-907 is a highly selective, orally active CB2 receptor inverse agonist and exerts anti-inflammatory effects in vivo. |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.
