Cat.No. | Name | Information |
---|---|---|
M7325 | Rimonabant Hydrochloride | Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity |
M6402 | ACPA | ACPA is a potent, selective CB 1 agonist. |
M5290 | (±)-SLV-319 | (±)-SLV319 (Ibipinabant) is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo. |
M4777 | Pregnenolone | Pregnenolone (3β -hydroxy-5-pregnen-20-one) is a powerful neurosteroid, and is the major precursor of various steroids, including steroids. Pregnenolone is a specific signaling inhibitor of cannabinoid CB1 receptor. |
M3282 | GW842166X | GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. |
M3266 | WIN 55212-2 mesylate | WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively. |
M2981 | Rimonabant | Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane. |
M2552 | CP 945598 | CP 945598 (Otenabant) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM. |
M2461 | BML-190 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
M2379 | AM251 | AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain. |
M2343 | AM-2201 | AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively. |
M2051 | CP 945598 hydrochloride | CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively). |
M2012 | AM1241 | AM1241 is a cannabinoid CB2 receptor selective agonist. |
M1907 | Org 27569 | Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor. |
M54860 | Vicasinabin | Vicasinabin (RG7774) is the potent agonist of cannabinoid receptor 2 (CB2). |
M54730 | INV-347 | INV-347 is a CB1R inverse agonist that can be used in studies related to obesity. |
M54196 | RVD-Hpα TFA | RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. |
M53236 | Hemopressin(human, mouse) TFA | Hemopressin TFA is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. |
M53235 | Hemopressin(rat) TFA | Hemopressin(rat) TFA is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. |
M53234 | Hemopressin(rat) | Hemopressin(rat) is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. |
M53233 | Pirnabine | Pirnabine is a cannabinoid receptor ligand. |
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