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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M11289 | Solabegron | Solabegron (GW 427353) is a selective agonist of β3 adrenergic receptor (β3-AR). The EC50 value of Solabegron was 22 nM in Chinese hamster ovarian cells. It can be used to study overactive bladder and irritable bowel syndrome. |
| M10994 | Higenamine hydrochloride | Higenamine hydrochloride (Norcoclaurine hydrochloride) is a beta2-AR agonist that is a key ingredient in the Aconitum of Chinese medicine used in heart failure-related studies. Higenamine hydrochloride (Norcoclaurine hydrochloride) has an anti-apoptotic effect. |
| M10684 | Phenylephrine | (R)-(-)-Phenylephrine is a selective α1- adrenergic receptor agonists, mainly used as decongestants. |
| M10654 | Ajmalicine (Raubasine) | Ajmalicine (Raubasine) is an adrenolytic agent which preferentially blocks alpha 1-adrenoceptor than alpha 2-adrenoceptor. Ajmalicine (Raubasine) is an reversible non-competitive nicotine receptor antagonist with an IC50 of 72.3 μM. |
| M10644 | L-765314 | L-765314 is a potent and selective antagonist of α1b adrenergic receptor with Ki of 5.4 nM and 2.0 nM for rat and human α1b adrenergic receptor, respectively. |
| M9329 | Fenoterol | Fenoterol is a β2 adrenoreceptor agonist with bronchodilator activity. |
| M9264 | Norepinephrine | Norepinephrine is generally considered to be a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. |
| M9201 | Vibegron | Vibegron is a potent and selective beta 3 adrenergic receptor agonist. |
| M8857 | Xylazine | Xylazine is a α2-adrenoceptor agonist, sedative, muscle relaxant. |
| M7848 | ICI 118,551 hydrochloride | ICI 118,551 hydrochloride is a highly selective β2-adrenoceptor antagonist. |
| M7743 | Dobutamine hydrochloride | Dobutamine hydrochloride is a selective β1-AR agonist. |
| M6887 | L-755,507 | L-755,507 is a very potent and selective β3 partial agonist. |
| M6291 | 5-Iodotubercidin | 5-IOdotubercidin (NSC 113939), an ATP analogue, is a potent inhibitor of adenosine kinase with an IC50 value of 26 nM. 5-IOdotubercidin (NSC 113939) initiates glycogen synthesis in isolated hepatocytes by activating phosphorylase and glycogen synthase. 5-IOdotubercidin (NSC 113939) also inhibits CK1, insulin receptor tyrosine kinase, phosphorylase kinase, PKA, CK2, PKC, and Haspin inhibitors. |
| M6061 | Xylometazoline HCl | Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM. |
| M6060 | Xylazine HCl | Xylazine is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant. |
| M6019 | Tizanidine HCl | Tizanidine hydrochloride is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. |
| M6000 | Terazosin HCl | Terazosin is a selective alpha-1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). It works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls. |
| M5999 | Terazosin HCl Dihydrate | Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH). |
| M5998 | Terazosin | Terazosin is a selective alpha1-antagonist used for treatment of symptoms of benign prostatic hyperplasia (BPH). |
| M5988 | Tamsulosin | Tamsulosin is a selective α1 receptor antagonist. |
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