Cat.No. | Name | Information |
---|---|---|
M2628 | Dexmedetomidine | Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects. |
M3057 | Terbutaline Sulfate | Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM. |
M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
M2420 | Labetalol hydrochloride | Labetalol hydrochloride is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors. |
M13893 | Labetalol | Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist. |
M5245 | Olodaterol | Olodaterol (BI1744) is a selective, long acting β2-adrenoceptor (β2-AR) agonist (EC50=0.1 nM and pKi= 9.14 for human β2-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis. |
M5239 | Batefenterol | Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively. |
M5116 | Formoterol Hemifumarate | Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease. |
M4821 | Vilanterol trifenatate | Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity. |
M4820 | Vilanterol | Vilanterol(GW642444, Veranterol) is a long-acting β2-AR agonist. PEC50 of β2-AR, β1-AR and β3-AR were 10.37, 6.98, 7.36, respectively. |
M4600 | Synephrine | Synephrine is an alkaloid from Citrus aurantium that is also an agonist of adrenoceptors. |
M4593 | Yohimbine-Hydrochloride | Yohimbine hydrochloride is an α2-adrenergic receptor antagonist. |
M4447 | 3-Hydroxy-4-methoxycinnamic-acid | Isoferulic acid (3-Hydroxy-4-methoxycinnamic acid) is a kind of cinnamic acid derivative with anti - diabetes activity. Isoferulic acid (3-hydroxy-4-methoxycinnamic acid) binds and activates α 1-adrenergic receptor (IC50=1.4 μM), Enhanced β -endorphin secretion (EC50=52.2 nM) and increased in vitro glucose use. Isoferulic acid also has activity against influenza virus. |
M3662 | Bambuterol hydrochloride | Bambuterol hydrochloride is an effective β -adrenergic receptor agonist. |
M3656 | Carteolol hydrochloride | Carteolol hydrochloride is a non-selective β -blocker used to study glaucoma. |
M3605 | Salbutamol hemisulfate | Salbutamol hemisulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM. |
M3551 | Silodosin | Silodosin is an α1-adrenoceptor antagonist with high uroselectivity. |
M3509 | Nebivolol | Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM. |
M3482 | Carvedilol | Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation. |
M3457 | Naftopidil | Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM. |
M3413 | Phenoxybenzamine hydrochloride | Phenoxybenzamine hydrochloride is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM. |
M3411 | Sotalol | Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM. |
M3408 | Maprotiline hydrochloride | Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant. |
M3372 | Clonidine hydrochloride | Clonidine hydrochloride is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg. |
M3330 | Phenylephrine hydrochloride | Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist. |
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