| Cat.No. | Name | Information |
|---|---|---|
| M3326 | Memantine hydrochloride | Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively. |
| M2079 | Chrysin | Chrysin is a naturally occurring flavone chemically extracted from the passion flowers Passiflora caerulea. |
| M9931 | ε-Viniferin | ε-Viniferin is a potent inhibitor for all the CYP family, with Ki values from 0.5-20 μM. |
| M9877 | Rhapontigenin | Rhapontigenin is a selective inactivator of cytochrome P450 1A1 with IC50 of 400 nM. |
| M9684 | (Rac)-Brassinazole | (Rac)-Brassinazole is a brassinosteroid (BR) biosynthesis inhibitor. |
| M9016 | Ezutromid | Ezutromid (BMN-195, SMT C1100) is a first-in-class oral bioavailable utrophin translational modulator with an EC50 value of 0.4 uM. |
| M8186 | Stiripentol | Stiripentol (BCX2600) can be used in the study of the third generation of antiepileptic drugs that enhance gaba energy neurotransmission. It's an inhibitor of cytochrome P450. |
| M7416 | TMS | TMS is a cytochrome P450 1B1 inhibitor. |
| M6451 | Apigenin | Apigenin is a competitive CYP2C9 inhibitor with a Ki of 2 μM. |
| M6389 | 1-Aminobenzotriazole (ABT) | 1-Aminobenzotriazole (ABT) is a cytochrome P450 inhibitor; inhibits 20-HETE synthesis. |
| M6318 | 17-ODYA | 17-ODYA is a lTB ω-hydroxylase inhibitor. |
| M6262 | Fadrozole | Fadrozole is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM. |
| M5650 | Fluconazole | Fluconazole is a fungal lanosterol 14 alpha-demethylase inhibitor, which thereby prevents the formation of ergosterol,used in the treatment and prevention of superficial and systemic fungal infections. |
| M5557 | Deferasirox | Deferasirox (ICL-670) is an iron chelator that causes iron loss that promotes BclxL downregulation and cell death. Deferasirox (ICL-670) also induced P450 3A4 and inhibited 2C8 and 1A2. |
| M5059 | Furafylline | Furafylline was a potent, non-competitive inhibitor of high affinity phenacetin O-deethylase activity of microsomal fractions of human liver, a reaction catalysed by P450IA2, with an IC50 value of 0.07 microM. |
| M4935 | 3-Cyano-7-ethoxycoumarin | 3-Cyano-7-ethoxycoumarin is a fluorogenic cytochrome P-450 substrate that generates blue fluorescent product upon enzyme cleavage. |
| M4722 | Amentoflavone | Amentoflavone is a natural biflavone compound which has anti-inflammatory, antioxidative and neuroprotective effects. |
| M4699 | Galangin | Galangin (Norizalpinin) is a regulator of arylhydrocarbon receptors and also inhibits the activity of CYP1A1. |
| M4595 | Isosilybin | Isosilybin (Isosilybinin) is a flavonoid from milk thistle; The IC50 value induced by CYP3A4 inhibition was 74 μM. |
| M4573 | Diosmetin | Diosmetin is a natural flavonoid that inhibits the activity of human CYP1A enzyme. The IC50 value of Diosmetin in HepG2 cells is 40 μM. |
| M4495 | Linderane | Linderane was isolated from Lindera Strychnifolia and is an irreversible inhibitor of Cytochrome P450 2C9 (CYP2C9). Linderane has been shown to relieve pain and cramps. |
| M4414 | Gentiopicrin | Gentiopicroside is a natural iridoid glycoside that can inhibit the activity of P450 with IC50 and Ki values of 61 µM and 22.8 µM for CYP2A6, respectively. Gentiopicroside has anti-inflammatory and antioxidant activities. |
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