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Cat.No.  Name Information
M9789 MS049 MS049 is a potent and selective inhibitor of PRMT4,6 with IC50 values of 34 nM and 43 nM, respectively.
M9788 PF-9366 PF-9366 is a novel inhibitor of human methionine adenosyltransferase 2A (Mat2A), with IC50 of 420 nM and Kd of 170 nM.
M9787 Aminopterin Aminopterin is a folic acid derivative used as a rodenticide that has been shown to be teratogenic, and a dihydrofolate reductase inhibitor used to treat rheumatoid arthritis and leukemia.
M9786 Nimustine hydrochloride Nimustine hydrochloride (ACNU) is a DNA cross-linking and DNA alkylating agent, which induces DNA replication blocking lesions and DNA double-strand breaks.
M9785 ML364 ML364 is a small molecule inhibitor of the deubiquitinase USP2 (IC50=1.1 μM) with potential anticancer activity.
M9784 Naloxegol oxalate Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
M9783 Sodium oxamate Sodium oxamate is a competitive LDHA (actate dehydrogenase A) inhibitor, it inhibits L(+)-lactate dehydrogenase and derails the entire gluconeogenic pathway.
M9782 Bucladesine calcium Bucladesine calcium is a cell-permeable cyclic AMP (cAMP) analog and selectively activates cAMP dependent protein kinase (PKA) by increasing the intracellular level of cAMP.
M9781 E7820 E7820 is a α2 integrin inhibitor which suppressing integrin alpha 2, a cell adhesion molecule expressed on endothelial cells.
M9780 Nigericin Nigericin is an antibiotic derived from Streptomyces hygroscopicus, it acts as an H+, K+, Pb2+ ionophore.
M9779 THZ531 THZ531 is a covalent CDK12 and CDK13 inhibitor with IC50 values of 158 nM and 69 nM, respectively.
M9778 Voxelotor Voxelotor (GBT440) is a hemoglobin S allosteric modulator.
M9777 4-Nitroimidazole 4-Nitroimidazole is an intermediate during the synthesis of 1-methyl-2,4,5-trinitro imidazole.
M9776 Darbufelone Darbufelone is a dual inhibitor of cellular PGF2α and LTB4 production, it is also a COX-2 inhibitor potentially for the treatment of rheumatoid arthritis.
M9775 Fluralaner Fluralaner inhibits γ-aminobutyric acid (GABA)-gated chloride channels (GABACls) and l-glutamate-gated chloride channels (GluCls).
M9774 Namodenoson Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity.
M9773 Triacetyl-ganciclovir Triacetyl-ganciclovir is related to ganciclovir, which may be used for toxicity studies and other analytical studies during commercial production of Ganciclovir.
M9772 CHIR-090 CHIR-090 is a very potent and selective LpxC inhibitor, it is also a two-step slow, tight-binding inhibitor of E. coli LpxC with Ki = 4.0 nM.
M9771 TRAP-6 TRAP-6 (Thrombin Receptor Activator Peptide 6) is a peptide fragment (residues 42-47) of protease-activated receptor 1 (PAR1) that acts as a PAR1 agonist.
M9770 Riboflavin phosphate sodium Riboflavin phosphate sodium is the phosphate sodium salt form of riboflavin, a water-soluble and essential micronutrient that is the principal growth-promoting factor in naturally occurring vitamin B complexes.
M9769 BP-1-102 BP-1-102 is a potent, orally bioavailable and selective STAT3 inhibitor with IC50 of 6.8 μM.
M9768 MK-7622 MK-7622 is a cholinesterase inhibitor, it is also a muscarinic M1 receptor positive allosteric modulator.
M9767 BAY1082439 BAY1082439 is an orally bioavailable inhibitor of the class I phosphoinositide 3-kinase (PI3K) alpha and beta isoforms with potential antineoplastic activity.
M9766 GNE-1858 GNE-1858 is a potent, and ATP-competitive inhibitor of hematopoietic progenitor kinase-1 (HPK1).
M9765 Dimethyl itaconate Dimethyl itaconate may be used in functionalization of isotactic poly(propylene).
M9764 MK-3903 MK-3903 is a potent and selective AMPK activator (EC50 = 8 nM).
M9763 AVN-492 AVN-492 is a potent and selective 5-HT6R antagonist, binds to 5-HT6R (Ki = 91 pM).
M9762 GNE-617 GNE-617 is a potent nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with IC50 value of 5nM.
M9761 AZD-5597 AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects against a range of cancer cell lines.
M9760 Chicken egg albumin Chicken egg albumin, or ovalbumin, is the major protein constituent of egg whites. Chicken egg albumin is a phosphorylated glycoprotein.
M9759 Recombinant Human BMP-4 Bone morphogenetic proteins (BMPs) constitute a subfamily within the TGF-β superfamily of structurally related signaling proteins.
M9758 Merimepodib Merimepodib, also known as VX-497, is an orally bioavailable IMPDH inhibitor with broad spectrum antiviral activities.
M9757 AC710 AC710 is a potent, selective and orally active platelet-derived growth factor receptor-family (PDGFR) kinase inhibitor with potential anticancer activity.
M9756 Pocapavir Pocapavir (also known as SCH-48973 and V-073) is a potent, selective anti-enterovirus agent.
M9755 CYC065 CYC065 (Fadraciclib) is an orally bioavailable inhibitor of cyclin dependent kinases 2 and 9 (CDK2/9) with IC50 values of 5 and 26 nM, respectively.
M9754 AZD5153 AZD5153 is a potent bivalent triazolopyridazine based Bromodomain and Extraterminal (BET) Inhibitor, with IC50 value of 5 nM.
M9753 PQR530 PQR530 is a highly potent dual pan-PI3K/mTORC1/2 inhibitor.
M9752 GDC-0077 GDC-0077 is a potent and selective PI3K inhibitor with IC50 of 0.038 nM.
M9751 VUF11207 fumarate VUF11207 fumarate is a CXCR7 agonist and a high-potency CXCR7 ligand (pKi=8.1).
M9750 Vipivotide tetraxetan Vipivotide tetraxetan (PSMA-617) is a potent prostate-specific membrane antigen (PSMA) inhibitor with Ki value of 0.37 nM, it is used to make 177Lu-PSMA-617, which is a radioactive molecule to fight cancer.
M9749 Cotadutide acetate Cotadutide acetate is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor, with EC50 values of 6.9 pM and 10.2 pM, respectively.
M9748 Lisinopril dihydrate Lisinopril Dihydrate is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks.
M9747 Lanifibranor Lanifibranor (IVA-337) is a peroxisome proliferator-activated receptors (PPAR) agonist, with EC50s of 1.5, 0.87 and 0.21 μM for human PPARα, PPARσ and PPARγ, respectively.
M9746 CU-CPT-8m CU-CPT8m is an antagonist of toll-like receptor 8 (TLR8) with Kd of 220 nM and IC50 of 67 nM in assay.
M9745 DIDS sodium salt DIDS sodium salt (MDL101114ZA) is a dual ABCA1 and VDAC1 inhibitor. DIDS sodium salt is also an anion transport inhibitor, which inhibits the ClC-Ka chloride channel and the bacterial ClC-ec1Cl-/H+ exchanger with IC50s of 100 μM and ~300 μM, respectively.
M9744 QM385 QM385 is a potent sepiapterin reductase (SPR) inhibitor with IC50 of 1.49 nM.
M9743 Tetramethylrhodamine ethyl ester perchlorate TMRE is a mitochondria specific dye (λex=549 nm, λem=575 nm).
M9742 CU-CPT-9a CU-CPT-9a is a potent TLR8 antagonist with IC50 of 0.5 nM, which that suppresses TLR8-mediated proinflammatory signaling in various cell lines and human primary cells.
M9741 CU-CPT9b CU-CPT9b is a potent and selective TLR8 inhibitor, with an IC50 of 0.7 nM.
M9740 Aurintricarboxylic acid Aurintricarboxylic acid is a nanomolar-potency, allosteric antagonist with selectivity towards αβ-methylene-ATP-sensitive P2X1Rs and P2X3Rs, with IC50 values of 8.6 nM and 72.9 nM for rP2X1R and rP2X3R, respectively.
M9739 GW-870086 GW-870086 is a glucocorticoid receptor agonist, with pIC50 of 10.1 in A549 cells expressing NF-κB.
M9738 LX2761 LX2761 is a locally acting SGLT1 and SGLT2 inhibitor in vitro with IC50 values of 2.2 nM and 2.7 nM for hSGLT1 and hSGLT2, respectively.
M9737 Pyrotinib Pyrotinib (SHR-1258) is an orally bioavailable, potent and selective EGFR/HER2 dual inhibitor, with IC50 values of 13 and 38 nM, respectively.
M9736 VHL Ligand 1 hydrochloride VHL Ligand 1 hydrochloride is the VH032-based VHL ligand used in the recruitment of the von Hippel-Lindau (VHL) protein.
M9735 ND-646 ND-646 is an allosteric inhibitor of the ACC enzymes ACC1 and ACC2 with IC50 values of 3.5 nM and 4.1 nM for recombinant hACC1 and hACC2, respectively.
M9734 4-Nitrophenyl N-acetyl-β-D-glucosaminide 4-Nitrophenyl N-acetyl-β-D-glucosaminide is a chromogenic substrate for N-acetyl-glucosaminidase.
M9733 Eliglustat tartrate Eliglustat tartrate is a potent and selective glucosylceramide synthase inhibitor with IC50 of 24 nM.
M9732 Gadopentetate dimeglumine Gadopentetate dimeglumine is used in combination with magnetic resonance imaging (MRI) to allow blood vessels, organs, and other non-bony tissues to be seen more clearly on the MRI.
M9731 Indoxyl sulfate potassium salt Indoxyl sulfate potassium salt (Potassium 1H-indol-3-yl sulfate) is a metabolite of tryptophan derived from dietary protein.
M9730 CTLA-4 inhibitor 1 CTLA-4 inhibitor 1 is a potent B7.1-CD28 interaction inhibitor with IC50 of 50 nM.
M9729 diABZI STING agonist 1 (compound 3) diABZI STING agonist-1 (compound 3) is a selective stimulator of interferon genes (STING) receptor agonist, with EC50s of 130, 186 nM for human and mouse, respectively.
M9728 Fluensulfone Fluensulfone is a new nematicide for chemical control of plant parasitic nematodes.
M9727 SBI-115 SBI-115 is a TGR5 (GPCR19) antagonist, it decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5.
M9726 GLX351322 GLX351322 is an NADPH oxidase 4 inhibitor, which inhibits hydrogen peroxide production from tetracycline inducible NOX4-overexpressing cells with IC50 of 5 uM.
M9725 Ponalrestat Ponalrestat is an orally active, selective and noncompetitive aldose reductase inhibitor.
M9724 JC-1 JC-1 is a fluorescent lipophilic carbocyanine dye used to measure mitochondrial membrane potential.
M9723 L-Kynurenine L-Kynurenine is an aryl hydrocarbon receptor agonist.
M9722 Tyrphostin AG528 Tyrphostin AG528 (Tyrphostin B66) is an inhibitor of EGFR and ErbB2 with IC50 values of 4.9 and 2.1 μM, respectively.
M9721 Qstatin Qstatin is a selective inhibitor of quorum sensing (QS) in vibrio species.
M9720 Aranidipine Aranidipine (MPC1304) is a calcium channel blocker which may positively affect ambulatory blood pressure. *This compound is unstable in solutions, freshly prepared is recommended.
M9719 ML367 ML367 is an inhibitor of ATAD5 stabilization.
M9718 DB07268 DB07268 is is a potent and selective JNK1 inhibitor, with IC50 of 9 nM.
M9717 Etosalamide Etosalamide (also known as Ethosalamide) is an antipyretic and analgesics agent.
M9716 AKOS B018304 AKOS B018304 is a potent inhibitor of chikungunya virus with low micro molar activity.
M9715 Erdafitinib Erdafitinib (JNJ-42756493) is a potent and selective orally bioavailable, pan FGFR inhibitor with potential antineoplastic activity.
M9714 CAY10465 CAY10465 is an analog of resveratrol acting as a potent and selective aryl hydrocarbon receptor agonist, with a Ki of 0.2 nM.
M9713 SJ000291942 SJ000291942 is a bone morphogenic protein (BMP) signaling activator.
M9712 Pyrocatechuic acid Pyrocatechuic acid (2,3-Dihydroxybenzoic acid) is a normal human benzoic acid metabolite found in plasma, and has increased levels after aspirin ingestion.
M9711 AG1557 AG1557 is a potent and ATP competitive inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase with pIC50 value of 8.194.
M9710 Roquinimex Roquinimex (LS2616; FCF89) is a quinoline-3-carboxamide with potential antineoplastic activity, which increases NK cell activity and macrophage cytotoxicity.
M9709 NSC228155 NSC228155 is an activator of EGFR, which binds to the extracellular region of EGFR and enhance tyrosine phosphorylation of EGFR.
M9708 Chymotrypsin α-Chymotrypsin is a serine peptidase and has 241 amino acid residues contained in three polypeptide chains (A chain-13 residues, B chain-131 residues, and C chain-97 residues) linked by disulfide bridges.
M9707 HAMNO (NSC111847) HAMNO (NSC111847) is a potent and selective inhibitor of replication protein A (RPA) interactions with proteins involved in the replication stress response.
M9706 Colivelin TFA Colivelin TFA is a brain penetrant neuroprotective peptide and a potent activator of STAT3.
M9705 CP-376395 CP-376395 is a CRF1-selective antagonist.
M9704 Shield-1 Shield-1 is a specific, cell-permeant and high-affinity ligand of FK506-binding protein-12 (FKBP), and reverses the instability by binding to mutated FKBP.
M9703 Hexadimethrine bromide Hexadimethrine bromide can be used to transfect mammalian cells with DNA. It can be used to increase the efficiency of lipofection transfections.
M9702 QX77 QX77 is a novel chaperone-mediated autophagy (cma) activator.
M9701 Diethylenetriaminepentaacetic acid Diethylenetriaminepentaacetic acid is a diethylenetriaminepentaacetic anhydride, which is a bifunctional chelating agent.
M9700 ML213 ML213 (CID-3111211) is a selective KV7.2 (KCNQ2) and KV7.4 (KCNQ4) channel opener, with EC50 values of 230 and 510 nM for KV7.2 and KV7.4, respectively.
M9699 KY-226 KY-226 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor with IC50 of 0.25 μM, which protects neurons from cerebral ischemic injury.
M9698 D-(+)-Trehalose dihydrate D-(+)-Trehalose is a non-reducing sugar, used as a food ingredient and pharmaceutical excipient.
M9697 Nicotinamide Riboside Chloride Nicotinamide Riboside Chloride is a pyridine-nucleoside form of vitamin B3 that functions as a precursor to nicotinamide adenine dinucleotide or NAD+.
M9696 Dihydroethidium Dihydroethidium (also known as Hydroethidine and PD-MY 003) is a cell-permeable blue fluorescent dye.
M9695 Ellipticine hydrochloride Ellipticine (NSC 71795) hydrochloride is a potent antineoplastic agent which inhibits DNA topoisomerase II activities.
M9694 Chlorhexidine Chlorhexidine is a disinfectant and topical anti-infective agent.
M9693 PDM2 PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist, with a Ki of 1.2 nM.
M9692 IAXO-102 IAXO-102 is a TLR4 antagonist, which inhibits TLR4 signalling.
M9691 JD-5037 JD-5037 is a cannabinoid-1 receptor blocker (CB1R antagonist) with IC50 of 1.5 nM.
M9690 PEO-IAA PEO-IAA is a novel potent auxin antagonist, which binds to transport inhibitor response 1/auxin signaling F-box proteins (TIR1/AFBs).

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