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Cat.No.  Name Information
M9218 ABBV-744 ABBV-744 is a BDII-selective BET bromodomain inhibitor that is used in the research of AML and metastic castration-resistant prostate cancer.
M9217 Givinostat Givinostat is an HDAC inhibitor with IC50s of 198 and 157 nM for HDAC1 and HDAC3, respectively.
M9216 VcMMAE VcMMAE is a anti-mitotic agent, monomethyl auristatin E (MMAE), linked via the lysosomally cleavable dipeptide, valine-citrulline (vc).
M9215 GK921 GK921 is a transglutaminase 2 (TGase 2) inhibitor.
M9214 GC7 Sulfate GC7 Sulfate is a deoxyhypusine synthase (DHPS) inhibitor.
M9213 Miridesap Miridesap is a ligand for serum amyloid P component (SAP) and intends to inhibit and dissociate SAP binding to amyloid fibrils and tangles.
M9212 Aramchol Aramchol is a cholesterol solubilizer that prevents gallstone formation in inbred mice.
M9211 BDP5290 BDP5290 is a potent inhibitor of both ROCK and MRCK with IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.
M9210 Ampicillin Ampicillin is an antibiotic against a variety of gram-positive and gram-negative bacteria.
M9209 SLx-2119 SLx-2119, also known as KD-025, is an orally bioavailable inhibitor of ROCK-II with IC50 of 105 nM.
M9208 PD0166285 PD0166285 is a potent Wee1 inhibitor and Chk1 inhibitor with IC50s of 24 nM and 72 nM, respectively.
M9207 Tributylammonium pyrophosphate Tributylammonium pyrophosphate
M9206 Biphenyl-4-sulfonyl chloride Biphenyl-4-sulfonyl chloride is a HDAC inhibitor with synthetic applications in palladium-catalyzed desulfitative C-arylation.
M9205 Glasdegib Glasdegib (PF-04449913) is a potent, orally bioavailable Smoothened (Smo) inhibitor with an IC50 of 4 nM.
M9204 Pam3CSK4 Pam3CSK4 is a Toll-like receptor 1/2 (TLR1/2) agonist.
M9203 Cytochalasin B Cytochalasin B is a cell-permeable mycotoxin binding to the barbed end of actin filaments, disrupting the formation of actin polymers, with Kd value of 1.4-2.2 nM for F-actin.
M9202 α-cyano-4-hydroxy-cinnamic acid α-CHCA is a classic monocarboxylate transporters (MCT) inhibitor.
M9201 Vibegron Vibegron is a potent and selective beta 3 adrenergic receptor agonist.
M9200 Ibodutant Ibodutant (MEN15596) is a potent and selective tachykinin NK2 receptor antagonist with a pKi of 10.1.
M9199 Avacopan Avacopan (CCX168) is a potent, selective and orally available complement 5a receptor inhibitor with an IC50 of 0.1 nM.
M9198 JTZ-951 Enarodustat (JTZ-951) is a potent and orally active factor prolyl hydroxylase inhibitor, with an EC50 of 0.22 μM.
M9197 Relugolix Relugolix, also known as TAK-385, is a luteinizing hormone-releasing hormone (LH-RH) receptor antagonist with an IC50 of 0.12 nM.
M9196 Elagolix sodium Elagolix Soidum is a potent, selective, orally active, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with Kd value of 54 pM.
M9195 Saroglitazar Saroglitazar is a novel peroxisome proliferator-activated receptor (PPAR) agonist with predominant PPARα and moderate PPARγ activity, with EC50 values of 0.65 pM and 3 nM in HepG2 cells, respectively.
M9194 Insulin (human) Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets.
M9193 Carbetocin Carbetocin is an agonist at peripheral oxytocin receptors.
M9192 Cholic acid Cholic acid is a major primary bile acid produced in the liver and usually conjugated with glycine or taurine. It facilitates fat absorption and cholesterol excretion.
M9191 Sodium pyrophosphate Sodium pyrophosphate is a colorless transparent crystalline chemical compound with the formula Na4P2O7.
M9190 β-Glycerol phosphate disodium salt pentahydrate β-Glycerol phosphate disodium salt pentahydrate is a potent protein phosphatase and tensin homolog (PTEN) inhibitor.
M9189 Eldecalcitol Eldecalcitol is an analog of 1,25-dihydroxyvitamin D3 that improves bone mineral density.
M9188 Clomethiazole Clomethiazole is a positive allosteric modulator at the barbiturate/picrotoxin site of the GABAA receptor.
M9187 p-Nitrophenol p-Nitrophenol (4-NP) can be used to prepare 4-aminophenol.
M9186 Bedaquiline Bedaquiline, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections.
M9185 Serlopitant Serlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist.
M9184 RO8994 RO8994 is a potent and selective spiroindolinone MDM2 inhibitor, with IC50 of 5 nM (HTRF binding assays) and 20 nM (MTT proliferation assays).
M9182 Gefapixant Gefapixant, also known as AF-219 or MK-7264, is a P2X3 receptor antagonist.
M9181 8-OH-DPAT 8-OH-DPAT (8-Hydroxy-DPAT) is a potent and selective 5-HT agonist, with a pIC50 of 8.19 for 5-HT1A.
M9180 Pyridostatin Trifluoroacetate Salt Pyridostatin Trifluoroacetate Salt is a G-quadruplexe stabilizer, with a Kd of 490 nM.
M9179 Nolatrexed HCl Nolatrexed HCl, also known as AG337, is a thymidylate synthase inhibitor.
M9178 GSK2292767 GSK2292767 is a potent and selective PI3Kδ inhibitor.
M9177 SirReal2 SirReal2 is a potent and selective Sirt2 inhibitor with IC50 of 140 nM.
M9176 DTP3 DTP3 is a selective GADD45β/MKK7 inhibitor, which inhibits cancer-selective NF-κB survival pathway.
M9175 Vacquinol-1 Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma cell death.
M9174 ARQ 621 ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor.
M9173 Cilengitide trifluoroacetate Cilengitide is a potent integrin inhibitor for αvβ3 and αvβ5 receptor with IC50 of 4.1 nM, 79 nM in cell-free assays respectively.
M9172 Emedastine Difumarate Emedastine Difumarate is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
M9171 Sodium succinate Sodium succinate is an important metabolite at the cross-road of several metabolic pathways.
M9170 Sodium Houttuyfonate Sodium Houttuyfonate is the active compound of the Houttuynia plant.
M9169 Thimerosal Thimerosal inhibits a wide range of thiol-dependent enzymes and proteins, such as PI3-kinase-dependent methionine synthetase, glutamate transport receptor, and Na++K+ dependence ATPase.
M9168 Berberine Berberine is an alkaloid in several plants with various biological functions, including insulin-sensitizing, anti-inflammatory, and anti-oxidant activity.
M9166 BMS-986142 BMS-986142 is a potent, selective, reversible BTK inhibitor, shows BTK IC50 = 0.5nM; human WB IC50 = 90 nM.
M9165 Rimegepant Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM.
M9164 Insulin(cattle) Insulin is a peptide hormone produced by beta cells of the pancreatic islets. The compound is unstable in solutions, freshly prepared is recommended.
M9163 Blasticidin S hydrochloride Blasticidin S HCl is a potent inhibitor of protein synthesis in both prokaryotic and eukaryotic cells. Blasticidin S hydrochloride is a nucleoside antibiotic isolated from Streptomyces griseochromogenes.
M9162 Triton x-100 Triton x-100 is a nonionic, non-denaturing detergent suitable for solubilization, isolation and purification of membrane protein complexes.It is chemically indistinguishable from Nonidet P-40.
M9161 NVP-ACC789 NVP-ACC789 is an inhibitor of human VEGFR-1, VEGFR-2 (mouse VEGFR-2), VEGFR-3 and PDGFR-β with IC50s of 0.38, 0.02 (0.23), 0.18, 1.4 μM, respectively.
M9160 BMS-582949 BMS-582949 is a potent and selective P38 mitogen-activated protein kinase (P38 MAPK) inhibitor with IC50 of 13nM.
M9159 Adjudin Adjudin (also known as AF-2364) is a potent Cl- channel blocker, with a superior mitochondria-inhibitory effect.
M9158 Dihexa Dihexa is an orally active, blood-brain barrier-permeable angiotensin IV analog, exhibits high affinity binding hepatocyte growth factor (HGF) with a Kd of 65 pM.
M9157 2-Phenylethyl isothiocyanate 2-Phenylethyl isothiocyanate is an NNK-induced lung tumorigenesis inhibitor.
M9156 Benzyl isothiocyanate Benzyl isothiocyanate is a naturally-occurring constituent of cruciferous vegetables with antibacterial properties.
M9155 Autophinib Autophinib is a novel potent autophagy inhibitor, inhibiting autophagy induced by starvation or Rapamycin with IC50 values of 90 and 40 nM, targeting the lipid kinase VPS34 with IC50 value of 19 nM in vitro.
M9154 Iodixanol Iodixanol is a nonionic hydrophilic compound commonly used as a contrast agent during coronary angiography.
M9153 ACY-738 ACY-738 is a potent, selective and orally-bioavailable HDAC6 inhibitor, with an IC50s of 1.7 nM.
M9152 CPI-637 CPI-637 is a potent and selective CBP/EP300 bromodomains inhibitor with IC50 of 0.03±0.01μM and 11.0±0.6 μM for CBP/EP300 and BRD4, respectively.
M9151 MI-503 MI-503 is a potent and selective Menin-MLL inhibitor with IC50 of 14.7 nM.
M9150 MI-463 MI-463 is a highly potent and orally bioavailable small molecule inhibitor of the Menin-MLL interaction, with an IC50 value of 15.3 nM.
M9149 MI-136 MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes.
M9148 SRT2104 SRT2104 is a selective brain-permeable activator of SIRT1.
M9147 Peficitinib Peficitinib (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor, with IC50s of 3.9, 5.0, 0.7 and 4.8 nM for JAK1, JAK2, JAK3 and Tyk2, respectively.
M9146 GSK1324726A GSK1324726A (I-BET726) is a highly selective inhibitor of BET family proteins with IC50 of 41 nM, 31 nM, and 22 nM for BRD2, BRD3, and BRD4, respectively.
M9145 MI-2 MI-2 (Menin-MLL Inhibitor 2) is a potent menin-MLL interaction inhibitor with IC50 of 446±28 nM.
M9144 PFI-3 PFI-3 is a selective chemical probe for SMARCA bromodomains, including SMARCA2, SMARCA4 and PB1(5) bromodomains with a Kd of 89 nM.
M9143 HPOB HPOB is a highly potent and selective inhibitor of histone deacetylase 6 (HDAC6) with IC50 of 56 nM, >30 fold less potent against other HDACs.
M9142 FLLL32 FLLL32 is a potent JAK2/STAT3 inhibitor with IC50 of <5 μM.
M9141 SGC-CBP30 SGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50 of 21 nM and 38 nM in cell-free assays, respectively.
M9140 Hinokitiol Hinokitiol (β-thujaplicin) is a component of essential oils isolated from Chymacyparis obtusa, reduces Nrf2 expression, and decreases DNMT1 and UHRF1 mRNA and protein expression, with anti-infective, anti-oxidative, and anti-tumor activities.
M9139 Benzamide Benzamide is an inhibitor of poly(ADP-ribose) polymerase with an IC50 of 3.3 μM.
M9138 Picolinamide Picolinamide is a strong inhibitor of poly (ADP-ribose) synthetase of nuclei from rat pancreatic islet cells.
M9137 Elamipretide Elamipretide, also known as MTP-131, is a cardiolipin peroxidase inhibitor and mitochondria-targeted peptide.
M9135 TAK-779 TAK-779 is a potent and selective nonpeptide antagonist of CCR5, with a Ki of 1.1 nM for CCR5.
M9134 Citreoviridin Citreoviridin is a mycotoxin and potent inhibitor of mitochondrial ATPase.
M9133 AKBA AKBA is an active triterpenoid compound from the extract of Boswellia serrata and Boswellia carteri Birdw, exerts anti-inflammatory therapeutic effects and noncompetitively inhibits 5-lipoxygenase, topoisomerase, and leukocyte elastase.
M9132 ABM-3627 ABM-3627, also known as Mutant EGFR inhibitor, is a selective and potent Mutated EGFR inhibitor.
M9131 ZK-756326 dihydrochloride ZK-756326 dihydrochloride is a potent, selective and non-peptide CCR8 chemokine receptor agonist.
M9130 LSN3154567 LSN3154567 (also known as Nampt-IN-1) is a potent and elective NAMPT inhibitor, inhibits purified NAMPT with an IC50 of 3.1 nM.
M9129 GNE-131 GNE-131 is a potent and selective inhibitor of human sodium channel NaV1.7, with an IC50 of 3 nM.
M9128 AZ31 AZ31 is a potent and highly selective ATM inhibitor.
M9127 ONO-8590580 ONO-8590580 is a GABAAα5 negative allosteric modulator which enhances long-term potentiation and improves cognitive deficits in preclinical models.
M9126 Ac-CoA Synthase Inhibitor 1 Ac-CoA Synthase Inhibitor 1 (also known as ACSS2 Inhibitor), an anti-virus agent, is a Ac-CoA Synthase Inhibitor.
M9125 Z-Guggulsterone Z-Guggulsterone is a mineralocorticoid, progesterone and glucocorticoid receptor antagonist (Ki values are 37, 224 and 252 nM respectively) and weak androgen receptor agonist (Ki = 315 nM).
M9124 DY268 DY268 is a potent FXR antagonist with IC50 of 7.5 nM.
M9123 MBX-4132 MBX-4132 is a member of a chemical class called oxadiazoles that inhibit trans translation by binding to the bacterial ribosome.
M9122 Tormentic Acid Tormentic Acid is a natural anti-inflammatory agent which inhibits production of tumor necrosis factor‑α (TNF‑α), interleukin 6 (IL‑6), and IL‑1β.
M9121 LY303511 hydrochloride LY303511 hydrochloride is a structural analogue of LY294002. LY303511 enhances TRAIL sensitivity of SHEP-1 neuroblastoma cells via hydrogen peroxide-mediated mitogen-activated protein kinase activation and up-regulation of death receptors.
M9120 Hexacosanoic acid Hexacosanoic acid is a long-chain fatty acid related to various diseases such as adrenoleukodystrophy (ALD), adrenomyeloneuropathy (AMN) and atherosclerosis.
M9119 JNJ-632 JNJ-632 is a potent HVV capsid assembly modulator and HBV replication inhibitor with EC50 of 100-200 nM for genotypes A-D.
M9118 Chebulinic acid Chebulinic acid is a potent natural inhibitor of M. tuberculosis DNA gyrase, also can inhibit SMAD-3 phosphorylation, inhibit H+ K+-ATPase activity.
M9117 W-54011 W-54011 is a potent, specific, and orally active CD88 (C5a receptor) antagonist, which inhibits the binding of 125I-labeled C5a to human neutrophils with a Ki value of 2.2 nM.
M9116 Atorvastatin Atorvastatin is an inhibitor of HMG-CoA reductase used as a cholesterol-lowering medication that blocks the production of cholesterol.


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