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Cat.No.  Name Information
M8927 VU-0155069 VU-0155069 is a potent and selective phospholipase D1 (PLD1) inhibitor.
M8926 Niraparib (MK-4827) tosylate Niraparib (MK-4827) tosylate is an excellent PARP1 and PARP2 inhibitor with IC50 of 3.8 and 2.1 nM, respectively.
M8925 LY3023414 LY3023414 is a selective ATP-competitive inhibitor of PI3Kα and mTOR, DNA-PK, and other class I PI3K family members.
M8924 Daprodustat Daprodustat (GSK1278863) is a novel, orally active HIF-prolyl hydroxylase inhibitor.
M8923 CCG215022 CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50 values of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, GRK5 and GRK1, respectively.
M8922 Brevianamide F Brevianamide F belongs to a class of naturally occurring 2,5-diketopiperazines.
M8921 Bentamapimod Bentamapimod, also known as AS602801, is an ATP-competitive JNK inhibitor with IC50 of 80 nM, 90 nM, and 230 nM for JNK1, JNK2, and JNK3, respectively.
M8920 BDA-366 BDA-366 is a small molecule antagonist that specifically binds the BCL2 BH4 domain, and has the ability to convert anti-apoptotic BCL2 into a pro-apoptotic death molecule.
M8919 BAY 59-3074 BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively.
M8918 BAY 1217389 BAY 1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM.
M8917 BAW2881 BAW2881 (NVP-BAW2881) is a potent and selective VEGFR2 inhibitor with activity to inhibit chronic and acute skin inflammation.
M8916 SU1498 SU 1498 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 (VEGFR2, aka FLK1; IC50 = 700 nM).
M8915 TP-0903 TP-0903 is a potent and selective AXL inhibitor with an IC50 value of 27 nM.
M8914 AZD6738 AZD6738 is an orally active, and selective ATR kinase inhibitor with IC50 of 1 nM.
M8913 Telotristat ethyl Telotristat ethyl, also known as LX1606, is an oral serotonin synthesis inhibitor or peripheral tryptophan hydroxylase (TPH) inhibitor.
M8912 ML-18 ML18 is Bombesin receptor subtype 3 (BRS-3) antagonist (IC50 = 4.8 μM).
M8911 GS967 GS967, also known as GS-458967, is a potent and selective blocker of cardiac late sodium current (late INa) with IC50 values of 0.13 and 0.21 μM for ventricular myocytes and isolated hearts, respectively.
M8910 Pamapimod Pamapimod is a novel p38 mitogen-activated protein kinase inhibitor, inhibited p38alpha and p38beta enzymatic activity, with IC50 values of 0.014 +/- 0.002 and 0.48 +/- 0.04 microM, respectively.
M8909 Miransertib Miransertib, also known as ARQ 092, is an oral activie, potent and selective AKT inhibitor with IC50 values: 5.0 nM (AKT1); 4.5 nM (AKT2); 16 nM (AKT3).
M8908 ASC-J9 ASC-J9, also known as GO-Y025 and Dimethylcurcumin, suppressesing castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors.
M8907 Acecainide HCl Acecainide HCl, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide.
M8906 Sematilide hydrochloride Sematilide (CK-1752) hydrochloride is a novel class III antiarrhythmic agent.
M8905 EBE-A22 EBE-A22 is a derivative of PD 153035, has no effect on EGF-R TK but maintains a high cytotoxic profile.
M8904 NIH-12848 NIH-12848 is a putative phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ) inhibitor.
M8903 SR-3029 SR-3029 is a potent and ATP competitive CK1δ and CK1ε inhibitor, with IC50s of 44 nM and 260 nM, respectively.
M8902 CVT-313 CVT-313 is a potent and selective inhibitor of CDK2 that prevents neointimal proliferation, which has an IC50 of 0.5 microM in vitro.
M8901 CHS-828 CHS-828 (GMX1778) is a potent and specific inhibitor of NAMPT with IC50 and Kd value of <25 nM and 120 nM, respectively.
M8900 TG6-10-1 TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2.
M8899 TH588 TH588 is a potent inhibitor of MTH1 (NUDT1) with an IC50 value of 5 nM.
M8898 APY0201 APY0201 is a potent and selective IL-12/23 inhibitor.
M8897 B-Raf-IN-1 B-Raf-IN-1 (MDK36057) is a potent b-Raf inhibitor with IC50 of 24 nM.
M8896 MDK36122 MDK36122, also known as H-PGDS Inhibitor I, is a Prostaglandin D Synthase (hematopoietic-type) Inhibitor with an IC50 Value of 0.7 nM.
M8895 MX69 MX69 is a dual inhibitor of MDM2 and XIAP that binds to MDM2 RING protein with binding Kd values of 2.34 μM.
M8894 GJ-103 GJ-103 is an active analog of the read-through compound GJ072.
M8893 Miriplatin Miriplatin is a chemotherapy agent which belongs to the class of alkylating agents.
M8892 Coluracetam Coluracetam (MKC-231) is a new choline uptake enhancer.
M8891 AI-1 AI-1 is a negative regulator of Nrf2.
M8890 Forchlorfenuron Forchlorfenuron is a synthetic cytokinin that inhibits septins and exhibits anti-parasitic, anticancer, and anti-angiogenic activities.
M8889 6-Methoxy-2-naphthoic acid 6-Methoxy-2-naphthoic acid is an NMDA receptor modulator.
M8888 Donepezil Donepezil(E 2020) is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM, respectively.
M8887 Btk inhibitor 2 Btk inhibitor 2 (BGB-3111) is a Brutons tyrosine kinase (BTK) inhibitor.
M8886 RAF709 RAF709 is a novel Raf kinase inhibitor with IC50 values of 0.4 and 1.5 nM for c-Raf and b-Raf, respectively.
M8885 Rafoxanide Rafoxanide is a novel allosteric inhibitor of SPAK and OSR1.
M8884 Febantel Febantel is a veteran anthelmintic (wormer) compound belonging to the chemical class of the benzimidazoles.
M8883 Ceforanide Ceforanide is a new cephalosporin with antibacterial activity and has a longer elimination half-life than any currently available cephalosporin.
M8882 Trelagliptin succinate Trelagliptin(SYR-472) succinate is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
M8881 Ombitasvir Ombitasvir is a potent inhibitor of the hepatitis C virus protein NS5A, with EC50s of 0.82 to 19.3 pM against HCV genotypes 1 to 5 and 366 pM against genotype 6a.
M8880 Paritaprevir Paritaprevir (ABT-450) is a potent non-structural protein 3/4A (NS3/4A) protease inhibitor with EC50 values of 1 and 0.21 nM for HCV 1a and 1b, respectively.
M8879 AOA hemihydrochloride Aminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T.
M8878 Inositol Nicotinate Inositol Nicotinate is a formulation of niacin, which is also called vitamin B3, an essential human nutrient.
M8877 Pixantrone Maleate Pixantrone dimaleate is a topoisomerase II inhibitor and DNA intercalator, with anti-tumor activity.
M8876 Itacitinib Itacitinib, also known as INCB39110 or INCB039110, is a potent JAK1 tyrosine kinase inhibitor.
M8875 ND-630 ND-630 is an ACC inhibitor of human ACC1 and ACC2 with IC50 values of 2.1 and 6.1 nM, respectively.
M8874 C188-9 C188-9 is a small-molecule STAT3 inhibitor, can block Th2 and Th17 cell expansion and cytokine production to prevent house dust mite (HDM)-induced airway inflammation and remodeling.
M8873 D-Luciferin potassium salt D-Luciferin potassium salt is the substrate of luciferases that catalyze the production of light in bioluminescent insects.
M8872 ZD 7114 hydrochloride ZD 7114 is a selective β3 adrenergic receptor agonist.
M8870 Zopolrestat Zopolrestat is an inhibitor of Aldose Reductase.
M8869 Zinterol hydrochloride Zinterol Hydrochloride is a β2 adrenergic receptor selective agonist.
M8868 Zerumbone Zerumbone is a TRAIL-induced apoptosis potentiator.
M8867 Zaragozic acid A trisodium salt Potent inhibitor, in vivo and in vitro, of mammalian, fungal and Saccharomyces cervisiae squalene synthase.
M8866 Zonisamide sodium salt Zonisamide sodium salt is an anti-epileptic.
M8865 Zimelidine dihydrochloride Serotonin transport blocker; antidepressant.
M8864 Zotepine Zotepine is an atypical antipsychotic.
M8863 YM 976 Phosphodiesterase type IV (PDE4) inhibitor.
M8862 YH439 YH439 is an aryl hydrocarbon receptor activator.
M8861 Xaliproden hydrochloride 5-HT1A serotonin receptor agonist; neuroprotectant.
M8860 X80 X80 is an inhibitor of xeroderma pigmentosum group A protein (XPA protein) required for the removal of all types of DNA lesions repaired by nucleotide excision repair Including both transcription coupled and global genomic nucleotide excision repair.
M8859 Xestospongin C Xestospongin C is a selective, reversible and membrane-permeable inhibitor of IP3 receptor.
M8858 XE-991 XE-991 is a KCNQ channel blocker; which is more potent than linopiridine.
M8857 Xylazine α2-adrenoceptor agonist, sedative, muscle relaxant.
M8856 WAY-100135 dihydrochloride WAY-100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM).
M8855 WR99210 WR99210 is a potent inhibitor of Plasmodium falciparum dihydrofolate reductase (DHFR), which is a major malarial drug target.
M8854 WAY-100635 maleate salt WAY-100635 maleate salt is a highly selective 5-HT1A serotonin receptor antagonist.
M8853 WIN 62,577 Non-peptide NK1 tachykinin receptor antagonist.
M8852 W-84 dibromide Potent allosteric modulator of M2 muscarinic acetylcholine receptors.
M8851 WAY 161503 hydrochloride The 5-HT2C receptors have been implicated in conditions including obesity, anxiety, depression, OCD, schizophrenia, migraine, nociception and erectile dysfunction.
M8850 WAY-213613 WAY-213613 is a selective GLT-1/EAAT2 inhibitor.
M8849 VO-OHpic trihydrate VO-OHpic trihydrate is a PTEN (phosphatase and tensin homologue deleted on chromosome 10) inhibitor.
M8848 VU0152100 Positive allosteric modulator of muscarinic choline receptor M4.
M8847 Valnoctamide Valproic acid (VPA) and derivatives such as valpromide and valnoctamide are anti-convulsant, mood stabilizing drugs, believed to function as indirect GABA agonists by inhibiting the transamination of GABA.
M8846 VU0238429 VU0238429 is a selective muscarinic acetylcholine receptor 5 (M5) positive allosteric modulator; causes leftward shift in acetylcholine potency.
M8845 Valpromide Valpromide (VPD) is a derivative of valproic acid (VPA) and is used as an antiepileptic drug.
M8844 Valeryl Salicylate Selective, irreversible COX-1 inhibitor.
M8843 Verrucarol Trichothecene mycotoxin that is a component of toxic mold.
M8842 Valinomycin K+-selective ionophoric cyclodepsipeptide; potassium ionophore which uncouples oxidative phosphorylation, induces apoptosis in murine thymocytes, inhibits NGF-induced neuronal differentiation and antagonizes ET-induced vasoconstriction.
M8841 Carboxytolbutamide In vivo tolbutamide metabolite.
M8840 Oxidized Nifedipine CYP3A4 nifedipine metabolite.
M8839 U-74389G Free radical lipid peroxidation inhibitor in cultured brain cells, monocytic THP1 cells, and LLC-PK1 cell layers.
M8838 UBP302 UBP302 is a selective GluR5 antagonist.
M8837 UK-78282 monohydrochloride UK-78282 blocks both Kv1.
M8836 U 18666A Inhibitor of cholesterol synthesis (inhibits desmosterol Δ24-reductase).
M8835 UA62784 Studies have also reported that UA62784 associates with tubulin at or near the colchicine-binding sites in cells and functions as a cytotoxic, microtubule inhibitor.
M8834 U-62066 Highly selective κ opioid receptor agonist; antitussive.
M8833 UK 14,304 UK 14,304 is an α2-adrenoceptor agonist.
M8832 U-69593 U-69593 is a selective κ opioid receptor agonist.
M8831 5-Methylurapidil Selective α1A-adrenoceptor antagonist; antihypertensive.
M8830 Triazolam Anxiolytic; ligand for the GABAA receptor benzodiazepine modulatory site.
M8829 Picropodophyllotoxin Picropodophyllotoxin is an insulin-like growth factor-I (IGF-I) receptor kinase inhibitor.
M8828 Tofisopam Ligand for the GABAA receptor benzodiazepine modulatory site.
M8827 Tyrphostin 51 EGFR tyrosine kinase inhibitor.


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