Free shipping on all orders over $ 500

Vasopressin Receptor Vasopressin Receptor

Inhibitors

Cat.No.  Name Information
M14067 Argipressin Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1.
M11457 Desmopressin Acetate Desmopressin is a synthetic octapeptide that is an analogue of the human hormone arginine vasopressin and has antidiuretic and procoagulant effects.
M11397 D[LEU4,LYS8]-VP TFA D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptors, with Ki values of 0.16 nM, 0.52 nM and 1.38 nM for rat, human and mouse V1b receptors, respectively. D[LEU4,LYS8]-VP TFA showed weak antidiuretic, vasopressor and oxytocin activity in vitro.
M11396 Terlipressin acetate Terlipressin acetate is a vasopressin analogue and a highly selective vasopressin V1 receptor agonist that reduces visceral blood flow and portal vein pressure and controls acute varicose rupture bleeding. Terlipressin acetate has anti-inflammatory and antioxidant effects and can be used to study hepatorenal syndrome and norepinephrine-resistant septic shock.
M11395 Lixivaptan Lixivaptan (VPA-985, WAY-VPA 985) is an orally active, selective vasopressin receptor V2 antagonist with IC50 values of 1.2 nM in humans and 2.3 nM in rats.
M11394 Felypressin Felypressin (PLV-2) is a non-catecholamine vasoconstrictor and a vasopressin 1 (Vasopressin 1) agonist. Felypressin is widely used in dental surgery.
M11393 RG7713 RG7713 (RO5028442) is a highly effective and selective brain-osmotic vasopressin 1A (V1a) receptor antagonist with Ki values of 1 nM (hV1a) and 39 nM (mV1a).
M10312 Argipressin Acetate Argipressin (Arg8-vasopressin) binds to vascular arginine vasopressin receptors V1, V2 and V3, and its Kd value against V1 in A7r5 rat aortic smooth muscle cells is 1.31 nM.
M7356 TASP 0390325 TASP0390325 is a potent and orally active arginine vasopressin receptor 1B (V1B receptor) antagonist with antidepressant and anxiolytic activities in rodents.
M6879 L-371,257 L-371,257 is a potent and selective oxytocin receptor antagonist.
M5431 Atosiban Atosiban(RW22164; Tractocile) is a nonapeptide, desamino-oxytocin analogue, and a competitive vasopressin/oxytocin receptor antagonist (VOTra). Atosiban inhibits the oxytocin-mediated release of inositol trisphosphate from the myometrial cell membrane.
M3480 Tolvaptan Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM for the inhibition of AVP-induced platelet aggregation.
M1917 Mozavaptan Mozavaptan (OPC-31260) is a selective vasopressin V2 receptor antagonist.



Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.