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D[LEU4,LYS8]-VP TFA

Cat. No. M11397

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D[LEU4,LYS8]-VP TFA  Structure
Size Price Availability Quantity
5mg USD 78  USD78 In stock
10mg USD 125  USD125 In stock
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Quality Control & Documentation
Biological Activity

D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptors, with Ki values of 0.16 nM, 0.52 nM and 1.38 nM for rat, human and mouse V1b receptors, respectively. D[LEU4,LYS8]-VP TFA showed weak antidiuretic, vasopressor and oxytocin activity in vitro.

Chemical Information
Molecular Weight 1026.24
Formula C47H67N11O11S2
CAS Number 42061-33-6 (free base)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Dariusz Sobolewski, et al. J Pept Sci. Analogues of AVP modified in the N-terminal part of the molecule with Pip isomers: TFA-catalysed peptide bond hydrolysis

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Keywords: D[LEU4,LYS8]-VP TFA supplier, Vasopressin Receptor, inhibitors, activators

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