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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M10492 | Ropivacaine | Ropivacaine is a member of the amino amide class of local anesthetics and acts as a potent sodium channel blocker. |
| M10470 | Raxatrigine hydrochloride | Raxatrigine hydrochloride (GSK-1014802 hydrochloride) is a selective, small-molecule, state-dependent Nav1.7 voltage-gated sodium channel blocker. |
| M10458 | Huwentoxin IV TFA | Huwentoxin IV TFA is a selective NaV1.7 channel blocker, which preferentially inhibits neuronal NaV1.7, 1.2 and 1.3 (IC50 values are 26, 150 and 338 nM respectively), compared to muscle subtypes NaV1.4 and 1.5 (IC50 = >10 μM). |
| M10113 | BI01383298 | BI01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5). |
| M9129 | GNE-131 | GNE-131 is a potent and selective inhibitor of human sodium channel NaV1.7, with an IC50 of 3 nM. |
| M9115 | PF-06869206 | PF-06869206 is an orally bioavailable selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1) with an IC50 of 380 nM. |
| M9103 | Eleclazine hydrochloride | Eleclazine HCl is a novel late Na+ current inhibitor, with IC50 value of 0.7 uM. |
| M9018 | Levobupivacaine | Levobupivacaine is a reversible neuronal sodium channel inhibitor. |
| M8988 | PF-05089771 | PF-05089771 is a selective Nav1.7 channel blocker that interacts with the voltage-sensor domain (VSD) of domain IV. |
| M8947 | PF-01247324 | PF-01247324 is a novel selective and orally bioavailable Nav 1.8 channel blocker with an IC50 of 196 nM for recombinant human Nav1.8 channel. |
| M8911 | GS967 | GS967, also known as GS-458967, is a potent and selective blocker of cardiac late sodium current (late INa) with IC50 values of 0.13 and 0.21 μM for ventricular myocytes and isolated hearts, respectively. |
| M8510 | Cariporide | Cariporide is a selective inhibitor of the Na+/H+ exchanger subtype 1 (NHE-1), also known as the Na+/H+ antiporter. |
| M8092 | PF-05089771 Tosylate | PF-05089771 Tosylate is a selective and potent inhibitor of the human voltage-gated sodium ion channel Nav1. |
| M7572 | Tenapanor | Tenapanor is an inhibitor of the Na+/H+ exchanger NHE3 with IC50 values of 5 and 10 nM against human and Rat NHE3, respectively. |
| M7552 | ETH2120 | Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the assay of sodium activity in blood, plasma, serum. etc. |
| M7520 | Brivaracetam | Brivaracetam (UCB 34714) is chemically related to levetiracetam (LEV, Keppra). It possesses a binding affinity for the synaptic vesicle protein 2A (SV2A) ten-fold above that of LEV and also shows an ability to inhibit Na+ channels. |
| M6085 | GSK-1014802 | CNV1014802(GSK-1014802) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor. |
| M6068 | Zonisamide | Zonisamide is an fDA-approved antiepileptic compound that blocks voltage-dependent sodium (+) and T-type calcium channels. |
| M6054 | Vinpocetine | Vinpocetine is a selective inhibitor of voltage-sensitive sodium channel for the treatment of stroke, vascular dementia and Alzheimer's disease. |
| M6006 | Tetracaine | Tetracaine is a topical local anesthetic for the eyes; works by interfering with entry of sodium ions into nerve cells. |
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