P-gp P-glycoprotein

Inhibitors

Cat.No.	Name	Information
M6706	Elacridar hydrochloride	Elacridar hydrochloride is a p-gp inhibitor.
M6267	Valspodar	Valspodar is a P-glycoprotein (P-gp) inhibitor widely used as overcoming multidrug resistance modulator.
M5881	Piperine	Piperine, a natural alkaloid isolated from Piper nigrum L, inhibits P-glycoprotein and CYP3A4 activities with an IC50 value of 61.94±0.054 μg/mL in HeLa cell.
M5609	Elacridar (GF120918)	Elacridar (GF120918) is a potent P-gp (MDR-1) and BCRP inhibitor.
M5294	Polyoxyethylene stearate	Polyoxyethylene stearate (POES) is a non-ionic emulsifying agent.
M4792	Sinapine-thiocyanate	Sinapine, an alkaloid derived from seeds of the cruciferous species, possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.
M1888	Tariquidar	Tariquidar (XR9576) is a selective, highly efficacious third generation P-glycoprotein (P-gp) inhibitor.
M1853	Biricodar	The pipecolinate derivative Biricodar (VX-710, Incel) is a clinically applicable modulator of P-glycoprotein (Pgp) with potential chemosensitizing activity.
M1845	LY335979 trihydrochloride	LY335979 (Zosuquidar trihydrochloride) is a selective Pgp (P-glycoprotein) inhibitor with a Ki of 59 nM.