| Cat.No. | Name | Information |
|---|---|---|
| M39035 | Roquefortine C | Roquefortine C, a fungal cyclopeptide isolated from Penicillium roquefortii, activates P-gp and also inhibits P450-3A and other haemoproteins. Roquefortine C has bacteriostatic activities against Gram-positive bacteria. |
| M14250 | Encequidar mesylate | Encequidar mesylate (HM30181 mesylate; HM30181A mesylate) is a competitive and potent P-glycoprotein inhibitor. |
| M14249 | Encequidar | Encequidar (HM30181; HM30181A) is a potent and selective inhibitor of P-glycoprotein. |
| M14248 | Dofequidar fumarate | Dofequidar fumarate(MS-209 fumarate), an orally active quinoline compound, has been reported to overcome MDR by inhibiting ABCB1/P-gp, ABCC1/MDR-associated protein 1, or both. |
| M11058 | Ganoderenic acid B | Ganoderenic acid B is a triterpenoid isolated from Ganoderma lucidum. Ganoderenic acid B effectively reverses ABCB1-mediated resistance of HepG2/ADM cells to Doxorubicin. |
| M7190 | Reversan | Reversan (CBLC4H10) is a selective MRP1 and P-gp inhibitor. |
| M6706 | Elacridar hydrochloride | Elacridar hydrochloride is a p-gp inhibitor. |
| M6267 | Valspodar | Valspodar is a P-glycoprotein (P-gp) inhibitor widely used as overcoming multidrug resistance modulator. |
| M5609 | Elacridar (GF120918) | Elacridar (GF120918) is a potent P-gp (MDR-1) and BCRP inhibitor. |
| M4792 | Sinapine-thiocyanate | Sinapine, an alkaloid derived from seeds of the cruciferous species, possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression. Sinapine thiocyanate is also an acetylcholinesterase (AChE) inhibitor. |
| M4298 | Tenacissoside-G | Tenacissoside G is a C21 steroid from the stem of Marsdenia tenacissima. Tenacissoside G reverses multidrug resistance in multidrug resistant cancer cells that overexpress p-glycoprotein (Pgp). |
| M3976 | (20S)-Protopanaxadiol | (20S)-Protopanaxadiol (aPPD) is one of the aglycones of the ginsenosides and has a wide range of pharmacological activities. |
| M1888 | Tariquidar | Tariquidar (XR9576) is a selective, highly efficacious third generation P-glycoprotein (P-gp) inhibitor. |
| M1853 | Biricodar | The pipecolinate derivative Biricodar (VX-710, Incel) is a clinically applicable modulator of P-glycoprotein (Pgp) with potential chemosensitizing activity. |
| M1845 | LY335979 trihydrochloride | LY335979 (Zosuquidar trihydrochloride) is a selective Pgp (P-glycoprotein) inhibitor with a Ki of 59 nM. *The compound is unstable in solutions, freshly prepared is recommended |
| M56553 | Zosuquidar | Zosuquidar (LY335979) is a P-glycoprotein (P-gp) inhibitor (Ki=59 nM). |
| M56552 | Tariquidar dimesylate | Tariquidar dimesylate (XR9576 dimesylate) is a P-glycoprotein (P-gp) inhibitor. |
| M56551 | Tariquidar dihydrochloride | Tariquidar dihydrochloride (XR9576 dihydrochloride) is a potent and specific inhibitor of P-glycoprotein (P-gp) with the high affinity (Kd=5.1 nM). |
| M54201 | Reversin 121 | Reversin 121 is a P-glycoprotein inhibitor. |
| M52753 | Reversin 205 | Reversin 205 ([Boc-Glu(Obzl)]2-Lys-Ome) is a P-glycoprotein (ABCB1) inhibitor. |
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