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Histamine Receptor Histamine Receptor

Inhibitors

Cat.No.  Name Information
M11287 JNJ-39758979 Jnj-39758979 is a selective, orally active, high-affinity histamine H4 receptor antagonist with Ki values of 12.5, 5.3 and 25 nM for human, mouse and monkey histamine H4 receptor, respectively. Jnj-39758979 antagonized histamine-induced cAMP inhibition with a pA2 of 7.9. Jnj-39758979 has good anti-inflammatory and antipruritic effects.
M10773 ABT-239 ABT-239 is a novel, highly effective, non-imidazole H3R antagonist and antagonist of TRPV1.
M10717 JNJ-5207852 JNJ-5207852 IS HISTAMINE H3 RECEPTORS ARE SELECTIVELY EFFECTIVE ANTAGONISTS, WHICH ARE H AGAINST RATS AND HUMANS3 receptors pKi the values are 8.9 and 9.24, respectively.
M10715 GSK189254A GSK189254A (GSK189254) is a novel and highly effective selective H3 receptor antagonist for H3 in humans and ratshpi
M10714 Pitolisant Pitolisant is a potent and selective non-imidazole recombinant hentistamine H3 receptor reversed agonist,Ki 0.16 nM.
M10391 Osthole Osthole (Osthol) is a natural antihistamine alternative with potential inhibition of histamine H1 receptor activity.
M9459 Mequitazine Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist.
M9290 S 38093 S 38093 is an inverse agonist at histamine H3 receptors, displays a moderate affinity for rat, mouse and human H3 receptors with Ki of 8.8, 1.44 and 1.2µM, respectively.
M9172 Emedastine Difumarate Emedastine Difumarate is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
M6111 Meta-Fexofenadine Meta -Fexofenadine (META -MDL-16455) is an impurity of Fexofenadine.
M5942 Roxatidine Acetate HCl Roxatidine Acetate HCl is a specific and competitive histamin H2-receptor antagonist, with IC50 of 3.2 μM, inhibits gastric acid secretion and ulcer formation.
M5921 Ranitidine HCl Ranitidine is a histamine H2-receptor antagonist, used to treat stomach or intestinal ulcers.
M5792 Mizolastine Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
M5752 Loratadine Loratadine is a histamine H1 receptor antagonist, used to treat allergies. Also acts as a selective inhibitor of B(0)AT2 with IC50 of 4 μM.
M5741 Lidocaine Lidocaine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM. Lidocaine (Lignocaine) also inhibits sodium channels involving complex voltage and using dependence
M5727 Lafutidine Lafutidine, a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion.
M5722 Ketotifen Fumarate Ketotifen Fumarate is a fumaric acid salt of ketotifen which is a H1-antihistamine and mast cell stabilizer.
M5692 Histamine Histamine is an organic nitrogenous compound involved in local immune responses as well as regulating physiological function in the gut and acting as a neurotransmitter.
M5638 Famotidine Famotidine is a histamine H2–receptor antagonist with IC50 of 0.6 mM, commonly used to treat heartburn, GERD, ulcers, and other digestive conditions.
M5615 Epinastine Epinastine(WAL801) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.



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