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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M11287 | JNJ-39758979 | Jnj-39758979 is a selective, orally active, high-affinity histamine H4 receptor antagonist with Ki values of 12.5, 5.3 and 25 nM for human, mouse and monkey histamine H4 receptor, respectively. Jnj-39758979 antagonized histamine-induced cAMP inhibition with a pA2 of 7.9. Jnj-39758979 has good anti-inflammatory and antipruritic effects. |
| M10773 | ABT-239 | ABT-239 is a novel, highly effective, non-imidazole H3R antagonist and antagonist of TRPV1. |
| M10717 | JNJ-5207852 | JNJ-5207852 IS HISTAMINE H3 RECEPTORS ARE SELECTIVELY EFFECTIVE ANTAGONISTS, WHICH ARE H AGAINST RATS AND HUMANS3 receptors pKi the values are 8.9 and 9.24, respectively. |
| M10715 | GSK189254A | GSK189254A (GSK189254) is a novel and highly effective selective H3 receptor antagonist for H3 in humans and ratshpi |
| M10714 | Pitolisant | Pitolisant is a potent and selective non-imidazole recombinant hentistamine H3 receptor reversed agonist,Ki 0.16 nM. |
| M10391 | Osthole | Osthole (Osthol) is a natural antihistamine alternative with potential inhibition of histamine H1 receptor activity. |
| M9459 | Mequitazine | Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist. |
| M9290 | S 38093 | S 38093 is an inverse agonist at histamine H3 receptors, displays a moderate affinity for rat, mouse and human H3 receptors with Ki of 8.8, 1.44 and 1.2µM, respectively. |
| M9172 | Emedastine Difumarate | Emedastine Difumarate is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. |
| M6111 | Meta-Fexofenadine | Meta -Fexofenadine (META -MDL-16455) is an impurity of Fexofenadine. |
| M5942 | Roxatidine Acetate HCl | Roxatidine Acetate HCl is a specific and competitive histamin H2-receptor antagonist, with IC50 of 3.2 μM, inhibits gastric acid secretion and ulcer formation. |
| M5921 | Ranitidine HCl | Ranitidine is a histamine H2-receptor antagonist, used to treat stomach or intestinal ulcers. |
| M5792 | Mizolastine | Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. |
| M5752 | Loratadine | Loratadine is a histamine H1 receptor antagonist, used to treat allergies. Also acts as a selective inhibitor of B(0)AT2 with IC50 of 4 μM. |
| M5741 | Lidocaine | Lidocaine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM. Lidocaine (Lignocaine) also inhibits sodium channels involving complex voltage and using dependence |
| M5727 | Lafutidine | Lafutidine, a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion. |
| M5722 | Ketotifen Fumarate | Ketotifen Fumarate is a fumaric acid salt of ketotifen which is a H1-antihistamine and mast cell stabilizer. |
| M5692 | Histamine | Histamine is an organic nitrogenous compound involved in local immune responses as well as regulating physiological function in the gut and acting as a neurotransmitter. |
| M5638 | Famotidine | Famotidine is a histamine H2–receptor antagonist with IC50 of 0.6 mM, commonly used to treat heartburn, GERD, ulcers, and other digestive conditions. |
| M5615 | Epinastine | Epinastine(WAL801) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis. |
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