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Pitolisant is a potent and selective non-imidazole recombinant hentistamine H3 receptor reversed agonist,Ki 0.16 nM.
| Molecular Weight | 295.85 |
| Formula | C17H26ClNO |
| CAS Number | 362665-56-3 |
| Solubility (25°C) | DMSO ≥ 60 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] No authors listed. CNS Drugs. Pitolisant
[2] No authors listed. Med Lett Drugs Ther. Pitolisant (Wakix) for narcolepsy
[4] Yvette N Lamb. CNS Drugs. Pitolisant: A Review in Narcolepsy with or without Cataplexy
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