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Cannabinoid Cannabinoid

Inhibitors

Cat.No.  Name Information
M7325 Rimonabant Hydrochloride Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity
M10720 A-836339 A-836339 is a selective agonist of the cb2 receptor and has little effect on the cb1 receptor.
M10652 Voacamine Voacamine is an indole alkaloid, exhibits potent cannabinoid CB1 receptor antagonistic activity. Voacamine also inhibits P-glycoprotein (P-gp) action in multidrug-resistant tumor cells.
M10218 (+)-Gallocatechin (+)-Gallocatechin is found notably in green tea, it has moderate affinity to the human cannabinoid receptor and acts as an antioxidant.
M9691 JD-5037 JD-5037 is a cannabinoid-1 receptor blocker (CB1R antagonist) with IC50 of 1.5 nM.
M9652 CB1-IN-1 CB1-IN-1 is a novel potent restricted CB1R antagonist with Ki of 0.3 nM and 21 nM for CB1R and CB2R, respectively.
M9136 Cannabidiol Cannabidiol is a GPR55 and weak CB1 antagonist with IC50s of 0.445 and 3.35 μM, it is also a CB2 receptor inverse agonist and inhibitor of anandamide uptake with IC50 of 27.5 μM.
M8985 LY2828360 LY2828360 is a novel potent, selective, and efficacious CB2 cannabinoid agonist.
M8919 BAY 59-3074 BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively.
M7325 Rimonabant Hydrochloride Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity
M7071 O-2050 O-2050 is a putative CB1 silent antagonist; displays mixed activity at CB receptors.
M6429 AM 630 AM 630 is a CB2 selective inverse agonist.
M5290 (±)-SLV-319 (±)-SLV319 (Ibipinabant) is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo.
M3282 GW842166X GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.
M3266 WIN 55212-2 mesylate WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively.
M2981 Rimonabant Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
M2552 CP 945598 CP 945598 (Otenabant) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
M2461 BML-190 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
M2343 AM-2201 AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.
M2051 CP 945598 hydrochloride CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively).
M2012 AM1241 AM1241 is a cannabinoid CB2 receptor selective agonist.



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