| Cat.No. | Name | Information |
|---|---|---|
| M7325 | Rimonabant Hydrochloride | Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity |
| M56149 | AEF0117 | AEF0117 is a signaling-specific inhibitor of the cannabinoid receptor 1 (CB1-SSi). |
| M55693 | HU-308 | HU-308 is a potent, selective agonist of the cannabinoid receptor CB2, with Ki values of 22.7nM and >10 mM for CB2 and CB1, respectively. HU-308 has anti-inflammatory and neuroprotective properties. HU-308 reduces liver damage in a hepatic ischemia/reperfusion injury model. |
| M45352 | Tetrahydrocannabivarin | Tetrahydrocannabivarin is an antagonist of cannabinoid receptors and may be used in studies related to type 2 diabetes. |
| M45350 | RVD-Hpα | RVD-Hpα is an alpha-hemoglobin-derived peptide containing three additional amino acids and a CB1 cannabinoid receptor agonist. In addition, RVD-Hpα is an orthosteric modulator of cannabinoid receptor 2 (CB2). |
| M25437 | Noladin ether | Noladin ether is a potent and selective agonist of cannabinoid CB1 receptor, with a Ki of 21.2 nM. |
| M21427 | CB1 agonist 1 | CB1 agonist 1 is an agonist of CB1. The pIC50 value of CB1 agonist 1 affinity with CB1 receptor was 5.7. CB1 agonist 1 can be used in the study of brain disorders. |
| M17348 | Olivetol | Olivetol is a naturally phenol found in lichens and produced by certain insects, acting as a competitive inhibitor of the cannabinoid receptors CB1 and CB2. Olivetol also inhibits CYP2C19 and CYP2D6 activity, with IC50s of 15.3 μM, 7.21 μM and Kis of 2.71 μM, 2.87 μM, respectively. |
| M14560 | Pregnenolone monosulfate | Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. |
| M13917 | Anandamide | Anandamide is an immune modulator in the central nervous system acts via not only cannabinoid receptors (CB1 and CB2) but also other targets (e.g., GPR18/GPR55). |
| M10720 | A-836339 | A-836339 is a selective agonist of the cb2 receptor and has little effect on the cb1 receptor. |
| M10719 | Yangonin | Yangonin has a high affinity for human recombinant cannabinoid CB1 receptors,IC50 and Ki 1.79 μM and 0.72 μM, respectively. |
| M10718 | TM38837 | TM38837 is an orally active, peripherally restricted cannabinoid receptor type 1 (CB1) receptor antagonist.TM38837 has limited penetration into the brain and minimizes or prevents CNS adverse effects. |
| M10652 | Voacamine | Voacamine is an indole alkaloid, exhibits potent cannabinoid CB1 receptor antagonistic activity. Voacamine also inhibits P-glycoprotein (P-gp) action in multidrug-resistant tumor cells. |
| M10218 | (+)-Gallocatechin | (+)-Gallocatechin is found notably in green tea, it has moderate affinity to the human cannabinoid receptor and acts as an antioxidant. |
| M9691 | JD-5037 | JD-5037 is a cannabinoid-1 receptor blocker (CB1R antagonist) with IC50 of 1.5 nM. |
| M9652 | CB1-IN-1 | CB1-IN-1 is a novel potent restricted CB1R antagonist with Ki of 0.3 nM and 21 nM for CB1R and CB2R, respectively. |
| M8985 | LY2828360 | LY2828360 is a novel potent, selective, and efficacious CB2 cannabinoid agonist. |
| M8919 | BAY 59-3074 | BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively. |
| M7613 | 2-Arachidonyl glycerol | 2-Arachidonyl glycerol is an endogenous cannabinoid and also an agonist at cannabinoid receptors. |
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