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TM38837 is an orally active, peripherally restricted cannabinoid receptor type 1 (CB1) receptor antagonist.TM38837 has limited penetration into the brain and minimizes or prevents CNS adverse effects.
| Molecular Weight | 617.51 |
| Formula | C30H25Cl2F3N4OS |
| CAS Number | 1253641-65-4 |
| Form | Solid |
| Solubility (25°C) | DMSO ≥ 20 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Robert J Chorvat. Bioorg Med Chem Lett. Peripherally restricted CB1 receptor blockers
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