Free shipping on all orders over $ 500

A-836339

Cat. No. M10720

All AbMole products are for research use only, cannot be used for human consumption.

A-836339 Structure
Size Price Availability Quantity
5mg USD 190  USD190 In stock
10mg USD 340  USD340 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

A-836339 is a selective agonist of the cb2 receptor and has little effect on the cb1 receptor.

Chemical Information
Molecular Weight 310.46
Formula C16H26N2O2S
CAS Number 959746-77-1
Solubility (25°C) DMSO ≥ 10 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] M Salaga, et al. Naunyn Schmiedebergs Arch Pharmacol . Highly selective CB 2 receptor agonist A836339 has gastroprotective effect on experimentally induced gastric ulcers in mice

[2] Rares-Petru Moldovan, et al. J Med Chem . Development of a High-Affinity PET Radioligand for Imaging Cannabinoid Subtype 2 Receptor

[3] Gin C Hsieh, et al. Br J Pharmacol . Central and peripheral sites of action for CB₂ receptor mediated analgesic activity in chronic inflammatory and neuropathic pain models in rats

[4] S McGaraughty, et al. Neuroscience . A CB(2) receptor agonist, A-836339, modulates wide dynamic range neuronal activity in neuropathic rats: contributions of spinal and peripheral CB(2) receptors

[5] Geraldine Pottier, et al. J Cereb Blood Flow Metab. PET imaging of cannabinoid type 2 receptors with [ 11 C]A-836339 did not evidence changes following neuroinflammation in rats

[6] Andrew G Horti, et al. Bioorg Med Chem. Synthesis and biodistribution of [11C]A-836339, a new potential radioligand for PET imaging of cannabinoid type 2 receptors (CB2)

[7] S McGaraughty, et al. Neuroscience. A CB(2) receptor agonist, A-836339, modulates wide dynamic range neuronal activity in neuropathic rats: contributions of spinal and peripheral CB(2) receptors

[8] Betty B Yao, et al. J Pharmacol Exp Ther. Characterization of a cannabinoid CB2 receptor-selective agonist, A-836339 [2,2,3,3-tetramethyl-cyclopropanecarboxylic acid [3-(2-methoxy-ethyl)-4,5-dimethyl-3H-thiazol-(2Z)-ylidene]-amide], using in vitro pharmacological assays, in vivo pain models, and 䲧璷Ỵ璸㧀璶羹瘬癳虸۪ř۪Ā�

Related Cannabinoid Products
UCM707 

UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of Anandamide.

SCH 336

SCH 336 is a potent, selective, inverse and orally active CB2 agonist.

JTE-907 

JTE-907 is a highly selective, orally active CB2 receptor inverse agonist and exerts anti-inflammatory effects in vivo.

LEI-101 

LEI-101 is a potent, selective, and orally bioavailable cannabinoid CB2 receptor agonist, with a pEC50 of 8 for hCB2, and a pKi of less than 4 for hERG.

AEF0117 

AEF0117 is a signaling-specific inhibitor of the cannabinoid receptor 1 (CB1-SSi).

  Catalog
Abmole Inhibitor Catalog




Keywords: A-836339 supplier, Cannabinoid, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.