Cat.No. | Name | Information |
---|---|---|
M9587 | NDI-091143 | NDI-091143 is a novel potent inhibitor of human ATP-citrate lyase with an IC50 of 2.1 nM (ADP-Glo assay), a Ki of 7.0 nM and a Kd of 2.2 nM. NDI-091143 inhibits ACLY catalysis allosterically, by stabilizing large conformational changes in the citrate domain that indirectly block the binding and recognition of citrate. |
M7737 | Concanamycin A (Folimycin) | Concanamycin A (Folimycin) is a macrolide antibiotic and a specific vacuolar type H+-ATPase (V-ATPase) inhibitor. |
M2294 | Brefeldin A | Brefeldin A is a lactone antibiotic and ATPase inhibitor for protein transport with IC50 of 0.2 μM in HCT 116 cells. Brefeldin A is also an autophagy and mitophagy inhibitor. Brefeldin A is a CRISPR/Cas9 activator. Brefeldin A inhibits HSV-1 and has anti-cancer activity. |
M1997 | Oligomycin A | Oligomycin A is an inhibitor of mitochondrial ATP synthase and uncoupler of oxidative phosphorylation. |
M10676 | Tegoprazan | Tegoprazan (CJ-12420, IN-A001, K-CAB, LXI-15028) is a potassium-competitive acid blocker and a potent, oral active and highly selective inhibitor of gastric H+/K+-ATPase that could control gastric acid secretion and motility, with IC50 values ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro. |
M10261 | Gboxin | Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma, inhibits the activity of F0F1 ATP synthase, with antitumour activity. |
M9719 | ML367 | ML367 is an inhibitor of ATAD5 stabilization. |
M9134 | Citreoviridin | Citreoviridin is a mycotoxin and potent inhibitor of mitochondrial ATPase. |
M8318 | KM91104 | KM91104 is a cell-permeable vacuolar ATPases (V-ATPase) inhibitor that specifically targets the V-ATPase a3-B2 subunits interaction. |
M5161 | Sodium orthovanadate | Sodium orthovanadate is an alkaline phosphatase and (Na,K)-ATPase inhibitor with IC50 of 10 μM. |
M3696 | Rostafuroxin | Rostafuroxin, a novel antihypertensive compound, acts as a selective inhibitor of srC-SH2 interaction with Na, K-ATPase activated by mutated adducin and Wabin in vivo. |
M2725 | Golgicide A | Golgicide A is a potent and rapidly reversible GBF1 inhibitor. |
M2474 | BTB06584 | BTB06584 is an IF1-dependent, selective inhibitor of the mitochondrial F1 Fo-ATPase. |
M56448 | Apoptolidin | Apoptolidin is a polyketide isolated from Nocardiopsis bacteria. |
M52778 | Transdermal Peptide Disulfide | Transdermal Peptide Disulfide (TD 1 Disulfide(peptide)) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly interacts with the C-terminus of ATP1B1. |
M52777 | SPAI-1 | SPAI-1 is a specific inhibitor for monovalent cation transporting ATPases. |
M42210 | Prilocaine acetate | Prilocaine acetate, an amino amide, is a Na/K-ATPase inhibitor. |
M42209 | Chamigrenol | Chamigrenol is a Na+/K+-ATPase inhibitor with an IC50 value of 15.9 μg/mL. |
M42161 | ZW290 | ZW290 is a compound to activate brown adipose tissue (BAT) thermogenic function. |
M42160 | ATP synthase inhibitor 2 TFA | ATP synthase inhibitor 2 TFA is a Pseudomonas aeruginosa (PA) ATP synthase inhibitor (IC50=10 μg/mL). |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.