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Sigma Receptor Sigma receptors

Cat.No.  Name Information
M10723 Ditolylguanidine Ditolylguanidine (1,3-Di-o-tolylguanidine) is a sigma receptor (σ1/σ2 receptor) agonist.
M10722 PRE-084 hydrochloride PRE-084 hydrochloride is a highly affinity selective σ1 agonist with an IC50 value of 44 nM in the sigma receptor detection.
M10721 Dimemorfan phosphate Dimemorfan phosphate is a potent agonist of sigma 1 receptor that is effective in suppressing cough.
M6496 BD 1063 dihydrochloride BD 1063 dihydrochloride is a selective σ1 ligand, putative antagonist.
M6495 BD 1047 dihydrobromide BD 1047 dihydrobromide is a σ 1 selective antagonist.
M6346 4-PPBP maleate 4-PPBP maleate is a specific σ ligand, NMDA antagonist.
M6344 4-IBP 4-IBP is a σ ligand, σ 1> σ 2.
M6203 Blarcamesine hydrochloride Blarcamesine hydrochloride is a Sigma-1 Receptor agonist with an IC50 of 860 nM.
M2991 SA 4503 dihydrochloride SA 4503 is a novel and selective opioid sigma1 receptor agonist with IC50 of 17.4 nM.
M2924 Pentoxyverine Citrate Pentoxyverine citrate is an orally active sigma-1 receptor agonist with Ki values of 41 nM for σ1, 894 nM for σ2, and 75 nM for σ1 in guinea pig brain membranes.Pentoxyverine citrate is also a muscarinic antagonist.
M2596 S1RA S1RA (E-52862) is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM), which showes good selectivity against σ2R (Ki > 1000 nM).
M2593 Siramesine hydrochloride Siramesine (Lu 28-179) hydrochloride is an effective sigma-2 receptor agonist. Siramesine has a nanomolar affinity for sigma-2 receptors (IC50=0.12 nM) and is 140 times more selective for sigma-2 receptors (IC50=17 nM). Siramesine has xC-system inhibitory activity associated with iron death.
M2592 Siramesine Siramesine (Lu 28-179) is a potent sigma-2 receptor agonist. Siramesine has a subnanomolar affinity for sigma-2 receptors (IC50=0.12 nM) and exhibits a 140-fold selectivity for sigma-2 receptors over sigma-1 receptors (IC50=17 nM). Siramesine triggers cell death through destabilisation of mitochondria, but not lysosomes.
M50236 ANAVEX 3-71 ANAVEX 3-71 is an orally active SIGMAR1 receptor agonist and M1-positive variant modulator for studies related to schizophrenia.
M45323 Blarcamesine Blarcamesine is a Sigma-1 receptor agonist and muscarinic receptor modulator with neuroprotective and antidepressant activity. In addition, Blarcamesine ameliorates neurological impairment in a mouse model of Rett syndrome.
M42707 AB10 AB10 is a selective S1R antagonist.
M42706 WLB-89462 WLB-89462 is a selective σ2 receptor ligand (Ki: 13 nM).
M42705 Siramesine fumarate Siramesine (Lu 28-179) fumarate is a potent sigma-2 receptor agonist.
M42704 Sigma-1 receptor antagonist 5 Sigma-1 receptor antagonist 5 and histamine H3 (hH3R, Ki=7.7 nM, IC50=215 nM).
M42703 AB21 AB21 is a potent and selective S1R antagonist with Kis of 13, 102 nM for S1R and S2R.




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