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CT1812 (Sigma-2 receptor antagonist 1) is an orally active and brain penetrant sigma-2 (σ-2) receptor antagonist with a Ki of 8.5 nM. CT1812 can be used for the research of Alzheimer’s disease.
| Molecular Weight | 431.59 |
| Formula | C24H33NO4S |
| CAS Number | 1802632-22-9 |
| Solubility (25°C) | DMSO 150 mg/mL |
| Storage | 2-8°C, protect from light |
[2] Ai-Fang Chen, et al. Sigma-2 Receptor as a Potential Drug Target
[4] Hayden R Schmidt, et al. The Molecular Function of σ Receptors: Past, Present, and Future
| Related Sigma Receptor Products |
|---|
| IPAG
IPAG is a potent sigma-1 receptor antagonist with a pKi of 4.3. |
| PB28 dihydrochloride
PB28 dihydrochloride, a cyclohexylpiperazine derivative, is a high affinity and selective sigma 2 (σ2) receptor agonist with a Ki of 0.68 nM. |
| (±)-PPCC hemioxalate
(±)-PPCC hemioxalate is a compound that has the ability to regulate the activity of the sigma-1 receptor. |
| (+)-Igmesine hydrochloride
(+)-Igmesine hydrochloride (JO1784) is an orally active and selective σ receptor ligand with neuroprotective and anti-amnesic activities. |
| ANAVEX 3-71
ANAVEX 3-71 is an orally active SIGMAR1 receptor agonist and M1-positive variant modulator for studies related to schizophrenia. |
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