| Cat.No. | Name | Information |
|---|---|---|
| M3629 | LY333531 hydrochloride | LY333531 hydrochloride competitively and reversibly inhibits PKCβI and PKCβII (IC50 values are 4.7 and 5.9 nM respectively). |
| M2066 | Staurosporine (AM-2282) | Staurosporine (AM-2282) is a potent ATP-competitive kinase inhibitor with IC50 of 0.7, 7, 8.5, 6, 20 nM for PKC, PKA,PKG, p60v-src tyrosine protein kinase, CaM kinase II, respectively. |
| M2850 | Midostaurin | Midostaurin (pkc412) is a multi-targeted kinase inhibitor, including PKCα/β/γ, Syk, Flk-1, Akt, PKA, c-Kit, c-Fgr, c-Src, FLT3, PDFRβ and VEGFR1/2 with IC50 ranging from 80-500 nM. |
| M4647 | Phorbol 12-myristate 13-acetate | Phorbol 12-myristate 13-acetate (PMA) is a dual SphK and protein kinase C (PKC) activator, increases the intracellular Ca2+ concentration ([Ca2+]i) in a dose-dependent manner, with an EC50 of 11.7 nM. |
| M5032 | Zoledronic acid monohydrate | Zoledronic acid monohydrate(CGP 42446; ZOL 446) is an activator of protein kinase C with apoptotic effects on multiple myeloma cell lines. It inhibited proliferation of human foetal osteoblastic cell line (hFOB) with an IC50 of 40 uM. |
| M2329 | Zoledronic acid | Zoledronic Acid (Zoledronate) is a third-generation bisphosphonate (BP), with potent anti-resorptive activity. Zoledronic Acid inhibits the differentiation and apoptosis of osteoclasts. Zoledronic Acid also has anti-cancer effects. |
| M2790 | K252a | K252a is an inhibitor of the BDNF receptor TrkB. K-252a inhibits protein kinase with IC50 values of 470 nM, 140 nM, 270 nM, and 1.7 nM for PKC, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase, respectively. K-252a is a potent inhibitor (IC50 of 3 nM) of the tyrosine protein kinase (TRK) activity of the NGF receptor gp140trk, the product of the trk protooncogene. |
| M54251 | Protein Kinase C (19-31) | Protein Kinase C (19-31), a peptide inhibitor of protein kinase C (PKC), is used as protein kinase C substrate peptide for testing the protein kinase C activity. |
| M54162 | Protein Kinase C (19-36) | Protein Kinase C (19-36) is a pseudosubstrate peptide inhibitor of protein kinase C (PKC), with an IC50 of 0.18 μM. |
| M53313 | [Ala113]MBP(104-118) | [Ala113]MBP(104-118) is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 28-62 μM. |
| M53312 | [Ala107]MBP(104-118) | [Ala107]MBP(104-118) is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 46-145 μM. |
| M53311 | Protein Kinase C (530-558) | Protein Kinase C (530-558), a peptide fragment of protein kinase C (PKC), is a potent PKC activator. |
| M53310 | Protein Kinase C (660-673) | Protein Kinase C (660-673) (PKC βII (660-673)) is the PKC βII V5 peptide with RACK1-binding affinity. |
| M53309 | PKCδ Peptide Substrate | PKCδ Peptide Substrate is an absolutely specific substrate for the δ-type of PKC, with a sequence corresponding to sequence 422-443 of murine eEF-1α and containing Thr-431. |
| M53308 | Myelin Basic Protein | Myelin Basic Protein (MHP4-14), a synthetic peptide comprising residues 4-14 of myelin basic protein, is a very selective PKC substrate (Km=7 μM). |
| M53307 | FKKSFKL-NH2 | FKKSFKL-NH2 is a protein kinase C-selective peptide. |
| M53306 | Z-Arg-SBzl | Z-Arg-SBzl is a substrate of both bovine and activated human protein C. |
| M53305 | PKCη pseudosubstrate inhibitor, myristoylated | PKCη pseudosubstrate inhibitor,myristoylated is cell permeable and can be used to study the mechanism of action of PKCη. |
| M53304 | [Ser25] Protein Kinase C (19-31) | [Ser25] Protein Kinase C (19-31) is a substrate of protein kinase C (PKC) (Km: 0.3 μM). |
| M53303 | pTH-Related Protein (1-40) (human, mouse, rat) | pTH-Related Protein (1-40) (human, mouse, rat) stimulates calcium uptake in rat intestinal cells through PTHR1 receptor and PKCα/β signaling pathways. |
| M53302 | [Ala9, 10, Lys11, 12] Glycogen Synthase (1-12) | [Ala9,10, Lys11,12] Glycogen Synthase (1-12) is a selective substrate for phosphorylation by protein kinase C (PKC). |
| M53301 | Protein Kinase C (19-35) Peptide | Protein Kinase C (19-35) Peptide is the PKC pseudosubstrate inhibitor/region. |
| M53300 | N-Myristoyl-Lys-Arg-Thr-Leu-Arg | N-Myristoyl-Lys-Arg-Thr-Leu-Arg is a protein kinase C (PKC) inhibitor with an IC50 value of 75 μM. |
| M53299 | Protein kinase C α peptide TFA | Protein kinase C (alpha) peptide (TFA) is a peptide of PKC-α. |
| M53298 | ɛPKC(85–92), Myristoylated | PKC(85–92),Myristoylated is a cell permeable myristic acid conjugated PKC peptide activator that enhances NO release in cultured human umbilical vein endothelial cells (HUVECs). |
| M53297 | Phosphate acceptor peptide | Phosphate acceptor peptide is a substrate for cAMP-dependent protein kinase (PKA). |
| M53296 | PKCβII Peptide Inhibitor I | PKCβII Peptide Inhibitor I is a PKCβII inhibitor. |
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