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UCN-02

Cat. No. M3799

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UCN-02 Structure
Size Price Availability
2mg USD 200 Out of stock
5mg USD 360 Out of stock
10mg USD 580 Out of stock
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Quality Control & Documentation
Biological Activity

UCN-02 is a stereoisomer of UCN-01. UCN-01 and UCN-02 showed the cytotoxic effect on the growth of HeLa S3 cells. UCN-02 is isolated as a minor co-metabolite of high staurosporine-producing strains of selected actinomycetes. Although less selective than its isomer UCN-01, UCN-02 exhibits comparable activity and probably acts by similar mechanisms.

Chemical Information
Molecular Weight 482.5
Formula C28H26N4O4
CAS Number 121569-61-7
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Takahashi I, et al. J Antibiot (Tokyo). UCN-01 and UCN-02, new selective inhibitors of protein kinase C. II. Purification, physico-chemical properties, structural determination and biological activities.

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Keywords: UCN-02 supplier, PKC, inhibitors, activators

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