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GCR Glucocorticoid Receptor

Cat.No.  Name Information
M3451 Hydrocortisone Hydrocortisone is a steroid hormone or glucocorticoid produced by the adrenal gland.
M21092 Vamorolone Vamorolone (VBP15) is the first orally active dissociative steroidal anti-inflammatory and membrane stabilizer. vamorolone improves myotonic dystrophy without side effects. vamorolone inhibits (NF-κB) inhibition and reduces the effects of hormones.
M13976 Desonide Desonide is a nonfluorinated corticosteroid anti-inflammatory agent used topically for dermatoses.
M13973 AZD9567 AZD9567 (compound 15) is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. Exhibits excellent efficacy in the streptococcal cell wall (SCW) reactivation model of joint inflammation.
M11555 Relacorilant Relacorilant is a selective, oral bioeffective glucocorticoid receptor antagonist (Ki of 7.2 nM in HepG2 TAT assay and 12,81.2 nM in rat, human and monkey glucocorticoid receptor in cell-based assay). Relacorilant can be used in studies of Cushing's syndrome.
M9739 GW-870086 GW-870086 is a glucocorticoid receptor agonist, with pIC50 of 10.1 in A549 cells expressing NF-κB.
M9545 Hydrocortisone Hemisuccinate Hydrocortisone hemisuccinate is an anti-inflammatory agent.
M7623 Beclomethasone Beclomethasone is a glucocorticoid receptor agonist with anti-inflammatory activity.
M6294 AZD-7594 AZD7594 is an inhaled, nonsteroidal, potent, and selective modulator of the glucocorticoid receptor (GR). It is being developed for once-daily treatment of chronic obstructive pulmonary disease and asthma, either alone or in combination with a bronchodilator.
M6281 (R)-Budesonide Budesonide is a GC steroid commonly used for the treatment of asthma and non-infectious rhinitis.
M5896 Prednisolone Acetate Prednisolone Acetate is a synthetic corticosteroid that is a particularly potent immunosuppressant.
M5695 Hydrocortisone acetate Hydrocortisone acetate is a corticosteroid, used to decrease swelling, itching, and pain that is caused by minor skin irritations or by hemorrhoids.
M5559 Deflazacort Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant.
M5535 Cortodoxone Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone).
M5534 Cortisone Cortisone is a 21-carbon steroid hormone. Cortisone is one of the main hormones released by the adrenal gland in response to stress.
M5533 Corticosterone Corticosterone (17-Deoxycortisol) is an orally active and adrenal cortex-produced glucocorticoid, which plays an important role in regulating neuronal functions of the limbic system. Corticosterone increases the Rab-mediated AMPAR membrane traffic via SGK-induced phosphorylation of GDI.
M5516 Ciclesonide Ciclesonide is a glucocorticoid used to treat obstructive airway diseases.
M5460 Betamethasone Betamethasone is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.
M5446 Beclometasone dipropionate Beclomethasone dipropionate is the precursor active molecule of Beclometasone and an orally effective glucocorticoid receptor agonist that acts through the glucocorticoid receptor to inhibit inflammation and hyperproliferation, and may be used in asthma-related studies.
M4882 AL 082D06 AL 082D06 is a selective non-steroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. There was no significant binding affinity for corticosteroids, androgens, estrogens and progesterone.




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