| Cat.No. | Name | Information |
|---|---|---|
| M9353 | N-Ethylmaleimide | N-Ethylmaleimide (NEM) is a cysteine protease inhibitor. |
| M3636 | Leupeptin hemisulfate | Leupeptin hemisulfate hemisulfate is the reversible inhibitor of lysosomal serine and cysteine proteinases; Leupeptin; inhibition of cathepsin B(Ki=6 nM), calpain(Ki=10 nM), trypsin (Ki=35 nM), plasmin (Ki=3.4 μM) and kallikrein (Ki=19 μM) had no effect on chymotrypsin, elastase, renin, or pepsin. |
| M2497 | Cathepsin Inhibitor 1 | Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively. |
| M1985 | Odanacatib | Odanacatib (MK-0822) is a potent and reversible covalent inhibitor of CathepsinK (CatK) with an IC50 of 0.2 nM/1 nM for human/rabbit cathepsin B, L, and S and is highly selective. |
| M14308 | SID 26681509 quarterhydrate | SID 26681509 quarterhydrate is a potent, reversible, competitive, and selective inhibitor of human cathepsin L with an IC50 of 56 nM. |
| M14307 | LY 3000328 | LY 3000328 is a potent and selective Cathepsin S (Cat S) inhibitor with IC50s of 7.7 and 1.67 nM for hCat S and mCat S, respectively. |
| M14306 | Cysteine Protease inhibitor hydrochloride | Cysteine Protease inhibitor hydrochloride is an inhibitor of cysteine protease. IC50 & Target: Cysteine Protease |
| M14305 | Cysteine Protease inhibitor | Cysteine Protease inhibitor is an inhibitor of cysteine protease. IC50 & Target: Cysteine Protease |
| M10280 | L006235 | L006235 (L235) is a potent, reversible cathepsin K inhibitor (IC50 = 0.25 nM) that displays > 4000-fold selectivity over cathepsins B, L and S. |
| M9318 | Chymostatin | Chymostatin is a chymotryptase-like serine proteases inhibitor, with Ki values of 9.36 and 13.1 nM for chymotrypsin and chymase, respectively. |
| M6236 | CA-074 Me | CA-074 Me is a membrane-permeable derivative of CA-074 and acts as an irreversible cathepsin B inhibitor. |
| M5288 | UK-371804 | UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). |
| M4767 | aurantiamide-acetate | Aurantiamide acetate is a selective and orally active cathepsin inhibitor isolated from Portulaca Oleracea L. Aurantiamide acetate has anti-inflammatory activity and can be used to study inflammatory diseases. |
| M3657 | Pepstatin A (Pepstatin) | Pepstatin A (Pepstatin) is a specific inhibitor of aspartic proteases produced by actinomycetes, which can inhibit hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease with IC50 values of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM, respectively. |
| M2823 | Loxistatin Acid(E-64C) | Loxistatin Acid (E-64C), a derivative of E-64, is an irreversible and membrane-permeant cysteine protease inhibitor. |
| M2600 | Balicatib | Balicatib is a potent and selective inhibitor of cathepsin K; 10-100-fold more potent in cell-based enzyme occupancy assays than against cathepsin B, L, and S. |
| M2376 | Aloxistatin | Aloxistatin (E64d) is an irreversible and membrane-permeable cysteine protease inhibitor. |
| M54370 | Z-Gly-Pro-Arg-AMC hydrochloride | Z-Gly-Pro-Arg-AMC hydrochloride a fluorescent trypsin and cathepsin K substrate. |
| M53923 | N-CBZ-Phe-Arg-AMC | N-CBZ-Phe-Arg-AMC (Z-FR-AMC) is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes. |
| M52672 | Ac-Glu-Asp(EDANS)-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Gly-Lys(DABCYL)-Glu-NH2 | Ac-Glu-Asp(EDANS)-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Gly-Lys(DABCYL)-Glu-NH2 is a cathepsin D substrate, that can be used for cathepsin D FRET assay. |
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