About 30 results found for searched term "RS-1" (0.01 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M1845 | LY335979 trihydrochloride | P-glycoprotein |
| Zosuquidar trihydrochloride; RS 33295-198 trihydrochloride | ||
| LY335979 (Zosuquidar trihydrochloride) is a selective Pgp (P-glycoprotein) inhibitor with a Ki of 59 nM. *The compound is unstable in solutions, freshly prepared is recommended | ||
| M2349 | (R)-Nepicastat hydrochloride | HCV Protease |
| RS-25560-198 HCl | ||
| (R)-Nepicastat hydrochloride, the R-enantiomer of Nepicastat hydrochloride, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors. | ||
| M2229 | Leflunomide | DHODH |
| HWA486; RS-34821; SU101 | ||
| Leflunomide (HWA486) is an inhibitor of dihydroorotate dehydrogenase with IC50 of 2.5 μM. | ||
| M2647 | DMH1 | ALK |
| dorsomorphin homolog 1 | ||
| DMH1 is a selective BMP receptor inhibitor with IC50 of 107.9 nM for ALK2, exhibiting no inhibition on AMPK, ALK5, KDR (VEGFR-2) or PDGFR. | ||
| M2662 | Efaproxiral Sodium | ROS |
| RSR13; NSC722758 | ||
| Efaproxiral sodium (RSR13 sodium) is a synthetic allosteric modifier of haemoglobin (Hb), decreases Hb-oxygen (O2) binding affinity and enhances oxygenation of hypoxic tumours. | ||
| M3267 | Nepicastat | Others |
| SYN117, RS-25560-197 | ||
| Nepicastat is a dopamine beta-hydroxylase inhibitor with IC50 of 8.5 ±0.8 and 9.0 ±0.8 nM for bovine and human, respectively. | ||
| M3363 | RS-127445 | 5-HT Receptor |
| MT500 | ||
| RS-127445 is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors. | ||
| M3416 | Mycophenolic acid | Immunology/Inflammation |
| Mycophenolate, RS-61443; MPA | ||
| Mycophenolic acid is an immunosuppressant agent used to prevent rejection in organ transplantation. | ||
| M3622 | Vernakalant | Potassium Channel |
| RSD-1235 | ||
| Vernakalant (RSD-1235) is an investigational mixed ion channel blocker, which can terminate acute atrial fibrillation (AF) in humans at 2 to 5 mg/kg and may be more atrial-selective than available agents. | ||
| M5794 | Moexipril HCl | ACE |
| RS-10085 | ||
| Moexipril HCl is a potent orally active nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor, used for the treatment of hypertension and congestive heart failure. | ||
| M6052 | Vernakalant HCl | Potassium Channel |
| RSD1235 hydrochloride | ||
| Vernakalant Hcl(RSD-1235) is an investigational mixed ion channel blocker that can terminate acute atrial fibrillation (AF) in humans at 2 to 5 mg/kg and may be more atrial-selective than available agents; in treatment of antiarrhythmic. | ||
| M6148 | RS-1 | CRISPR/Cas9 |
| RS-1 is a RAD51-stimulatory compound, which increases the DNA binding activity of RAD51. It is an HDR(homology-directed repair) enhancer. | ||
| M6997 | MRS 1220 | Others |
| MRS 1220 is a highly potent, selective hA 3 antagonist. | ||
| M6998 | MRS 1334 | Adenosine Receptor |
| MRS 1334 is a potent, highly selective hA 3 antagonist. | ||
| M6999 | MRS 1706 | Adenosine Receptor |
| MRS 1706 is a potent and selective A 2B inverse agonist. | ||
| M7000 | MRS 2179 tetrasodium salt | P2 Receptor |
| MRS 2179 tetrasodium salt is a selective P2Y 1 antagonist. | ||
| M7001 | MRS 2219 | Others |
| MRS 2219 is a potentiates P2X 1-mediated responses. | ||
| M7217 | RS 100329 hydrochloride | Others |
| RS 100329 hydrochloride is a potent, subtype-selective α 1A antagonist. | ||
| M7218 | RS102895 hydrochloride | CCR |
| RS 102895 HCl | ||
| RS102895 hydrochloride is a cCR2b chemokine receptor antagonist. | ||
| M7219 | RS 127445 hydrochloride | Others |
| MT 500 | ||
| RS 127445 hydrochloride is a selective, high affinity 5-HT 2B antagonist. | ||
| M7220 | RS 17053 hydrochloride | Others |
| RS 17053 hydrochloride is a α 1A antagonist. | ||
| M7221 | RS 23597-190 hydrochloride | Others |
| RS 23597-190 hydrochloride is a 5-HT 4 antagonist. | ||
| M7223 | RS 45041-190 hydrochloride | Others |
| RS 45041-190 hydrochloride is a high affinity I 2 ligand. Highly selective. | ||
| M7225 | RS 56812 hydrochloride | Others |
| RS 56812 hydrochloride is a 5-HT 3 partial agonist. | ||
| M7906 | MRS1845 | Calcium Channel |
| MRS-1845 | ||
| MRS1845 is a selective store-operated calcium (SOC) channel inhibitor with an IC50 of 1.7 μM. | ||
| M7908 | MRS 1523 | Adenosine Receptor |
| MRS1523 | ||
| MRS 1523 is a selective A3 adenosine receptor antagonist in the rat. | ||
| M7915 | MRS 1191 | Adenosine Receptor |
| MRS1191 | ||
| MRS 1191 is putative A3 adenosine receptor antagonist, highly selective for human A3 receptor vs human A1 receptor. | ||
| M8446 | RSC133 | HDAC |
| RSC-133 | ||
| RSC133 is an epigenetic modulator that effectively enhances reprogramming of human somatic cells and maintenance of human stem cell pluripotency. | ||
| M9045 | ARS-1620 | Ras |
| ARS-1620 is an atropisomeric selective KRAS-G12C inhibitor with desirable pharmacokinetics. | ||
| M9046 | ARS-1323 | Ras |
| ARS-1323 is a novel inhibitor of mutant K-ras G12C. | ||
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