About 30 results found for searched term "IAP" (0.161 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2259 | Biapenem | Antibiotic |
| L-627; LJC 10627; CLI 86815 | ||
| Biapenem is a new parenteral carbapenem antibacterial agent with a broad spectrum of in vitro antibacterial activity. | ||
| M3320 | Quetiapine Fumarate | 5-HT Receptor |
| Quetiapine hemifumarate | ||
| Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor. | ||
| M1565 | Quetiapine sulfoxide | 5-HT Receptor |
| Quetiapine sulfoxide; Quetiapine S-oxide | ||
| Quetiapine sulfoxide is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2. | ||
| M1564 | Quetiapine Sulfone | 5-HT Receptor |
| Quetiapine Sulfone is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2. | ||
| M5297 | Telacebec | Anti-infection |
| Q-203; Q 203; IAP6 | ||
| Telacebec (Q203; IAP6) is a midazopyridine amide compound. Q203 is active against Mycobacterium tuberculosis H37Rv with an MIC50 of 2.7 nM in culture broth medium. | ||
| M6332 | Triapine | DNA/RNA Synthesis |
| 3-AP; PAN-811; OCX191 | ||
| Triapine (3-AP; PAN-811) is a potent inhibitor of the M2 subunit of ribonucleotide reductase (RR), and it is a potent radiosensitizer. | ||
| M10814 | Eliapixant | P2 Receptor |
| BAY 1817080 | ||
| Eliapixant (BAY 1817080) is an effective and selective P2X3 receptor antagonist.IC50 The value is 8 nM. Eliapixant can be used in the study of refractory chronic cough. | ||
| M13874 | Quetiapine | 5-HT Receptor |
| ICI204636 | ||
| Quetiapine (ICI204636) is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. | ||
| M14263 | Tertiapin-Q | Potassium Channel |
| Tertiapin-Q is a highly selective blocker of GIRK1/4 heterodimer and ROMK1 (Kir1.1). | ||
| M16689 | 3,8''-Biapigenin | Flavonoids |
| 3,8''-Biapigenin | ||
| M17223 | Myrciaphenone A | Phenols |
| Myrciaphenone A | ||
| M20665 | Tiapride Hydrochloride | Dopamine Receptor |
| Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain and is used to treat a variety of neurological and psychiatric disorders. | ||
| M28346 | XIAP/cIAP1 antagonist-1 | IAP |
| XIAP/cIAP1 antagonist-1 is a potent and orally active XIAP/cIAP1 antagonist with EC50s of 5.1 nM and 0.32 nM for XIAP and cIAP1, respectively. XIAP/cIAP1 antagonist-1 inhibits the tumor growth in dose-dependent manner in vivo. | ||
| M29923 | Tiaprofenic acid | COX |
| Tiaprofenic acid is an orally active nonsteroidal anti-inflammatory agent (NSAID) with anti-inflammatory and analgesic potency. Tiaprofenic acid inhibits prostaglandin synthesis by suppressing cyclo-oxygenase (COX). Tiaprofenic acid can be used in the treatment of rheumatic diseases. | ||
| M30154 | Diaplasinin | PAI-1 |
| PAI-749 | ||
| Diaplasinin (PAI-749) is a plasminogen activator inhibitor-1 (PAI-1) inhibitor with IC50 of 295 nm. Antithrombotic efficacy. | ||
| M30523 | Tiaprost | Prostaglandin Receptor |
| Iliren | ||
| Tiaprost is a prostaglandin F2α (PGF2α) analogue. | ||
| M31316 | DiaPep277 | Immunology/Inflammation |
| DiaPep 277 | ||
| DiaPep277 is a peptide containing 24 amino acids based on residues 437 to 460 of Heat Shock Protein 60 (HSP60) for studies related to the immune system in type 1 diabetes. | ||
| M40914 | Rivulariapeptolides 1155 | Serine/Threonine Protease |
| Rivulariapeptolides 1155 is a potent serine protease inhibitor with IC50 values of 41.84 nM, 4.94 nM, and 56.54 nM for chymotrypsin, elastase, and proteinase K, respectively. | ||
| M40915 | Rivulariapeptolides 988 | Serine/Threonine Protease |
| Rivulariapeptolides 988 is a potent and selective serine protease inhibitor with IC50 values of 95.46 nM, 15.29 nM and 85.50 nM for tryptic coagulase, elastase and proteinase K, respectively. | ||
| M40916 | Rivulariapeptolides 1185 | Serine/Threonine Protease |
| Rivulariapeptolides 1185 is a potent and selective serine protease inhibitor with IC50 values of 13.17 nM, 23.59 nM, and 55.26 nM for tryptic coagulase, elastase, and proteinase K, respectively. | ||
| M40917 | Rivulariapeptolides 1121 | Serine/Threonine Protease |
| Rivulariapeptolides 1121 is a potent and selective serine protease inhibitor with IC50 values of 35.52 nM, 13.24 nM, and 48.05 nM for tryptic coagulase, elastase, and proteinase K, respectively. | ||
| M41092 | Diaporthein B | Antibiotic |
| Diaporthein B is one of the most highly oxidized pimarane diterpenes. | ||
| M41350 | MDM2/XIAP-IN-2 | Mdm2 |
| MDM2/XIAP-IN-2 is a dual inhibitor of murine double minute 2 (MDM2) and X-linked inhibitor of apoptosis protein (XIAP). | ||
| M41354 | MDM2/XIAP-IN-3 | Mdm2 |
| MDM2/XIAP-IN-3 is a dual MDM2/XIAP inhibitor. | ||
| M43085 | MDM2/XIAP-IN-1 | Others |
| MDM2/XIAP-IN-1 is an orally active inhibitor of dual MDM2/XIAP. | ||
| M43686 | Salviaplebeiaside | Others |
| Salviaplebeiaside is a phenolic substance can be isolated from the aerial part of Vitex negundo var. | ||
| M44935 | Microgrewiapine A | AChR/AChE |
| Microgrewiapine A is an antagonist of nAChR. | ||
| M53276 | Amylin (IAPP), feline | Others |
| Amylin (IAPP), feline is a 37-amino acid polypeptide from feline. | ||
| M58137 | L-Sepiapterin | Metabolite/Endogenous Metabolite |
| Sepiapterin | ||
| L-Sepiapterin (Sepiapterin) is a precursor of the endothelial nitric oxide synthase (eNOS) cofactor tetrahydrobiopterin (BH4). L-Sepiapterin improves endothelial dysfunction in small mesenteric arteries from db/db mice, and induces angiogenesis. | ||
| M55453 | Quetiapine-d8 fumarate | 5-HT Receptor |
| Quetiapine-d8 fumarate | ||
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