About 9 results found for searched term "98-10-2" (0.198 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M20427 | Benzenesulfonamide | Carbonic Anhydrase |
| Benzenesulphonamide, Benzosulfonamide, Phenyl sulfonamide, Benzene sulfonamide | ||
| Benzenesulfonamide ia an inhibitor of carbonic anhydrases. | ||
| M54491 | Fmoc-Lys(Biotin)-OH | Amino Acid Derivatives |
| Fmoc-Lys(Biotin)-OH is a lysine derivative. | ||
| M2428 | BAF312 | S1P Receptor |
| Siponimod | ||
| BAF312 (Siponimod) is a next-generation S1P receptor modulator, selective for S1P1 and S1P5 receptors with EC50 of 0.39 nM and 0.98 nM, exhibits >1000-fold selectivity over S1P2, S1P3 and S1P4 receptors. | ||
| M2578 | RITA | p53 |
| NSC 652287 | ||
| RITA (NSC 652287) is a MDM2 inhibitor and DNA damage agent for A498 (wild type) and TK-10 (mutation) cell lines with a GI50 of 17 nM and 32 nM, respectively. | ||
| M5403 | Alvimopan dihydrate | Opioid Receptor |
| LY 246736 dihydrate; ADL 8-2698 dihydrate | ||
| Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). | ||
| M6876 | L-161982 | Prostaglandin Receptor |
| L161982 | ||
| L-161982 is a EP4 receptor antagonist that is selective over all other members of the prostanoid receptor family (Ki values are 0.024, 0.71, 1.90, 5.10, 5.63, 6.74, 19 and 23 μM for human EP4, TP, EP3, DP, FP, IP, EP1 and EP2 receptors respectively). L-161982 completely blocks PGE2-induced ERK phosphorylation and cell proliferation of HCA-7 cells. | ||
| M27813 | CM398 | Sigma Receptor |
| CM398 is a highly selective, orally active sigma-2 receptor ligand (Ki=0.43 nM), with high sigma-1/sigma-2 selectivity rato (1000-fold). CM398 shows notable affinity for dopamine (Ki=32.90 nM) and serotonin transporters (Ki=244.2 nM). CM398 shows promising anti-inflammatory analgesic effects in the formalin model of inflammatory pain in mice. | ||
| M29694 | CHIR-98023 | GSK-3 |
| CHIR-98023 is a potent, selective and reversible inhibitor of GSK3, with IC50s of 10 nM and 6.7 nM for GSK3α and GSK3β, respectively. CHIR-98023 can improve insulin action and glucose metabolism. | ||
| M49546 | ENMD-1198 | Microtubule |
| ENMD-1198 (IRC-110160), an orally active microtubule destabilizing agent, is a 2-methoxyestradiol analogue with antiproliferative and antiangiogenic activity. | ||
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