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R406 besylate

Cat. No. M14916

All AbMole products are for research use only, cannot be used for human consumption.

R406 besylate Structure
Synonym:

R406 benzenesulfonate; Tamatinib

Size Price Availability Quantity
5mg USD 130  USD130 In stock
10mg USD 195  USD195 In stock
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Quality Control & Documentation
Biological Activity

R406 is an orally available and competitive Syk/FLT3 inhibitor for ATP binding with a Ki of 30 nM, potently inhibits Syk kinase activity in vitro with an IC50 of 41 nM, measured at an ATP concentration corresponding to its Km value. R406 reduces immune complex-mediated inflammation. R406 also inhibits Lyn (IC50=63 nM) and Lck (IC50=37 nM).

Chemical Information
Molecular Weight 628.63
Formula C22H23FN6O5.C6H6O3S
CAS Number 841290-81-1
Solubility (25°C) DMSO ≥ 61 mg/mL
Storage 2-8°C, dry, sealed
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  Catalog
Abmole Inhibitor Catalog




Keywords: R406 besylate, R406 benzenesulfonate; Tamatinib supplier, Syk, inhibitors, activators

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