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OP-3633 is a potent and selective steroidal glucocorticoid receptor (GR) antagonist with an IC50 of 29 nM, with inhibition of GR transcriptional activity. OP-3633 exhibits low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism.
| Molecular Weight | 445.64 |
| Formula | C30H39NO2 |
| CAS Number | 2102494-14-2 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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