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MLS1082 

Cat. No. M30806

All AbMole products are for research use only, cannot be used for human consumption.

MLS1082  Structure

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Quality Control & Documentation
Biological Activity

MLS1082 is a pyrimidone-based D1-like dopamine receptor positive allosteric modulator, with an EC50 of 123 nM for DA-stimulated G protein signaling.

Chemical Information
Molecular Weight 385.46
Formula C24H23N3O2
CAS Number 883958-36-9
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Kathryn D Luderman, et al. Bioorg Med Chem Lett. Development of pyrimidone D1 dopamine receptor positive allosteric modulators

[2] Kathryn D Luderman, et al. Mol Pharmacol. Identification of Positive Allosteric Modulators of the D1 Dopamine Receptor That Act at Diverse Binding Sites

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  Catalog
Abmole Inhibitor Catalog




Keywords: MLS1082  supplier, Dopamine Receptor, inhibitors, activators

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