Free shipping on all orders over $ 500

Ecopipam

Cat. No. M27812

All AbMole products are for research use only, cannot be used for human consumption.

Ecopipam Structure
Synonym:

SCH 39166

Price and Availability

For this product's availability, delivery time and price, please email [email protected] directly or click the "Inquiry Now" button below.


Quality Control & Documentation
Biological Activity

Ecopipam (SCH 39166) is a potent, selective and orally active antagonist of dopamine D1/D5 receptor, with Kis of 1.2 nM and 2.0 nM, respectively. Ecopipam shows more than 40-flod selectivity over D2, D4, 5-HT, and α2a receptor (Ki=0.98, 5.52, 0.08, and 0.73 μM, respectively). Ecopipam can be used for the research of schizophrenia and obesity.

Chemical Information
Molecular Weight 313.82
Formula C19H20ClNO
CAS Number 112108-01-7
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Donald L Gilbert, et al. Pediatrics. Ecopipam for Tourette Syndrome: A Randomized Trial

[2] Jessica Frey, et al. Curr Neurol Neurosci Rep. Tourette Syndrome Treatment Updates: a Review and Discussion of the Current and Upcoming Literature

[3] Kallol K Set, et al. Curr Probl Pediatr Adolesc Health Care. Tourette syndrome in children: An update

[4] Andrew Billnitzer, et al. Neurotherapeutics. Current Management of Tics and Tourette Syndrome: Behavioral, Pharmacologic, and Surgical Treatments

[5] Gerald A Maguire, et al. Ann Clin Psychiatry. Ecopipam as a pharmacologic treatment of stuttering

Related Dopamine Receptor Products
AJ-76

AJ-76 ((+)-AJ 76; (1S,2R)-AJ 76) is a dopamine autoreceptor antagonist.

A-412997 

A-412997 is a selective Dopamine D4 agonist with Ki values of 12 and 7.9 nM for the rat and human receptors.

SKF 81297 

SKF 81297 is a potent and selective dopamine D1 receptor agonist.

GBR 12783 

GBR 12783 is a specific, potent and selective dopamine uptake inhibitor that inhibits the [3H]dopamine uptake by rat and mice striatal synaptosomes with IC50s of 1.8 nM and 1.2 nM, respectively.

RMI-61140 

RMI-61140 is an orally active neuroleptics.

  Catalog
Abmole Inhibitor Catalog




Keywords: Ecopipam, SCH 39166 supplier, Dopamine Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.